# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4110365 | BDBM205421 | Ki | = | 13 | nM | ALA3887929 | 7.89 | 363864 | nM | Homo sapiens | |
2. | ALA4110365 | BDBM205421 | EC50 | = | 358 | nM | ALA3887928 | 6.45 | 363855 | nM | Homo sapiens | |
3. | ALA4110365 | BDBM205421 | F | = | 80.1 | % | ALA4355768 | % | ||||
4. | ALA4110365 | BDBM205421 | Vdss | = | 2.49 | L/Kg | ALA4355765 | L.kg-1 | ||||
5. | ALA4110365 | BDBM205421 | t1/2 | = | 1.95 | hr | ALA4355762 | hr | ||||
6. | ALA4110365 | BDBM205421 | CL | = | 25.7 | ml/min.kg | ALA4355760 | mL.min-1.kg-1 | ||||
7. | ALA4110365 | BDBM205421 | AUC/dose | = | 2.26 | uM.hr.kg/mg | ALA4355759 | uM.hr.kg/mg | ||||
8. | ALA4110365 | BDBM205421 | EC50 | = | 358 | nM | ALA4355755 | 6.45 | nM | Rattus norvegicus | ||
9. | ALA4110365 | BDBM205421 | Ki | = | 11 | nM | ALA4355754 | 7.96 | nM | Homo sapiens | ||
10. | ALA4110365 | BDBM205421 | Ki | > | 10000 | nM | ALA4355756 | nM | Homo sapiens |