| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4127309 | 23b | IC50 | = | 0.17 | nM | ALA4119717 | 9.77 | nM | |||
| 2. | ALA4127309 | 23b | IC50 | = | 24.6 | nM | ALA4119718 | 7.61 | nM | |||
| 3. | ALA4127309 | 23b | Ratio IC50 | = | 23 | ALA4119719 | ||||||
| 4. | ALA4127309 | 23b | TGI | 0 | ALA4119720 | Active | ||||||
| 5. | ALA4127309 | 23b | F | = | 7.4 | % | ALA4119729 | % | Rattus norvegicus | |||
| 6. | ALA4127309 | 23b | Tmax | = | 0.25 | hr | ALA4119728 | hr | Rattus norvegicus | |||
| 7. | ALA4127309 | 23b | Cmax | = | 0.48 | uM | ALA4119727 | nM | Rattus norvegicus | |||
| 8. | ALA4127309 | 23b | AUC | = | 0.33 | uM.hr | ALA4119726 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 9. | ALA4127309 | 23b | t1/2 | = | 0.32 | hr | ALA4119725 | hr | Rattus norvegicus | |||
| 10. | ALA4127309 | 23b | Vdss | = | 1.47 | L/Kg | ALA4119724 | L.kg-1 | Rattus norvegicus | |||
| 11. | ALA4127309 | 23b | CL | = | 74.66 | ml/min.kg | ALA4119723 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 12. | ALA4127309 | 23b | AUC | = | 0.88 | uM.hr | ALA4119722 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 13. | ALA4127309 | 23b | TGI | 0 | ALA4119721 | Active |
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