# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | DS88790512 | DS88790512 | solubility | = | 630 | ug ml-1 | ALA4122837 | ug.mL-1 | ||||
2. | DS88790512 | DS88790512 | solubility | = | 730 | ug ml-1 | ALA4122836 | ug.mL-1 | ||||
3. | DS88790512 | DS88790512 | Fu | > | 30 | % | ALA4122835 | |||||
4. | DS88790512 | DS88790512 | Stability | = | 96 | % | ALA4122834 | % | ||||
5. | DS88790512 | DS88790512 | F | = | 50 | % | ALA4122833 | % | Mus musculus | |||
6. | DS88790512 | DS88790512 | Vd | = | 24 | L/Kg | ALA4122832 | L.kg-1 | Mus musculus | |||
7. | DS88790512 | DS88790512 | CL | = | 180 | ml/min.kg | ALA4122831 | mL.min-1.kg-1 | Mus musculus | |||
8. | DS88790512 | DS88790512 | t1/2 | = | 2.9 | hr | ALA4122830 | hr | Mus musculus | |||
9. | DS88790512 | DS88790512 | AUC | = | 1000 | nM.hr | ALA4122829 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
10. | DS88790512 | DS88790512 | Cmax | = | 260 | nM | ALA4122828 | nM | Mus musculus | |||
11. | DS88790512 | DS88790512 | IC50 | > | 300 | uM | ALA4122826 | nM | Homo sapiens | |||
12. | DS88790512 | DS88790512 | IC50 | > | 100 | uM | ALA4122825 | nM | Homo sapiens | |||
13. | DS88790512 | DS88790512 | IC50 | = | 0.011 | uM | ALA4122824 | 7.96 | nM | Homo sapiens |