| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4128368 | 14j | F | = | 22.08 | % | ALA4257189 | % | ||||
| 2. | ALA4128368 | 14j | MRTlast | = | 5.01 | hr | ALA4257188 | hr | ||||
| 3. | ALA4128368 | 14j | %AUCextra | = | 25.87 | % | ALA4257187 | % | ||||
| 4. | ALA4128368 | 14j | AUC | = | 2453 | ng.hr/ml | ALA4257186 | ng.hr.mL-1 | ||||
| 5. | ALA4128368 | 14j | AUClast | = | 1646 | ng.hr/ml | ALA4257185 | ng.hr.mL-1 | ||||
| 6. | ALA4128368 | 14j | t1/2 | = | 5.3 | hr | ALA4257184 | hr | ||||
| 7. | ALA4128368 | 14j | Tmax | = | 3.33 | hr | ALA4257183 | hr | ||||
| 8. | ALA4128368 | 14j | Cmax | = | 271 | ng/ml | ALA4257182 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 9. | ALA4128368 | 14j | IC50 | > | 10000 | nM | ALA4257181 | nM | Homo sapiens | |||
| 10. | ALA4128368 | 14j | IC50 | = | 9360 | nM | ALA4257180 | 5.03 | nM | Homo sapiens | ||
| 11. | ALA4128368 | 14j | IC50 | = | 1000 | nM | ALA4257179 | 6.00 | nM | Homo sapiens | ||
| 12. | ALA4128368 | 14j | IC50 | = | 316 | nM | ALA4257178 | 6.50 | nM | Homo sapiens | ||
| 13. | ALA4128368 | 14j | IC50 | = | 5 | nM | ALA4257176 | 8.30 | nM | Homo sapiens | ||
| 14. | ALA4128368 | 14j | IC50 | = | 1500 | nM | ALA4257177 | 5.82 | nM | Homo sapiens | ||
| 15. | ALA4128368 | 14j | F | = | 22.1 | % | ALA4124025 | % | Cavia porcellus | |||
| 16. | ALA4128368 | 14j | AUC | = | 2452 | ng.hr/ml | ALA4124024 | ng.hr.mL-1 | Cavia porcellus | |||
| 17. | ALA4128368 | 14j | t1/2 | = | 5.25 | hr | ALA4124023 | hr | Cavia porcellus | |||
| 18. | ALA4128368 | 14j | Tmax | = | 3.33 | hr | ALA4124022 | hr | Cavia porcellus | |||
| 19. | ALA4128368 | 14j | Cmax | = | 271 | ng/ml | ALA4124021 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Cavia porcellus | ||
| 20. | ALA4128368 | 14j | AUC | = | 815 | ng.hr/ml | ALA4124020 | ng.hr.mL-1 | Cavia porcellus |
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