| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4159390 | 1 | INH | 0 | ALA4149796 | Dose-dependent effect | % | Homo sapiens | ||||
| 2. | ALA4159390 | 1 | INH | = | 79 | % | ALA4149795 | % | Homo sapiens | |||
| 3. | ALA4159390 | 1 | Ki | = | 0.69 | uM | ALA4149762 | 6.16 | nM | Homo sapiens | ||
| 4. | ALA4159390 | 1 | solubility | = | 1.1 | uM | ALA4149760 | nM | ||||
| 5. | ALA4159390 | 1 | Papp | < | 2.2 | 10'-6 cm/s | ALA4149759 | 10'-6 cm/s | ||||
| 6. | ALA4159390 | 1 | CLH(app) | > | 560 | microL/min/mg | ALA4149758 | mL.min-1.g-1 | ||||
| 7. | ALA4159390 | 1 | logD | = | 3.9 | ALA4149757 | ||||||
| 8. | ALA4159390 | 1 | IC50 | = | 4.3 | uM | ALA4149756 | 5.37 | nM | Homo sapiens | ||
| 9. | ALA4159390 | 1 | IC50 | > | 27 | uM | ALA4149755 | nM | Homo sapiens | |||
| 10. | ALA4159390 | 1 | IC50 | = | 5.4 | uM | ALA4149754 | 5.27 | nM | Homo sapiens | ||
| 11. | ALA4159390 | 1 | IC50 | = | 1.9 | uM | ALA4149753 | 5.72 | nM | Homo sapiens | ||
| 12. | ALA4159390 | 1 | IC50 | = | 0.15 | uM | ALA4149752 | 6.82 | nM | Homo sapiens | ||
| 13. | ALA4159390 | 1 | IC50 | = | 0.46 | uM | ALA4149751 | 6.34 | nM | Homo sapiens |
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