| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA137386 | 2a (E-isomer) | Ratio Ki | = | 32.2 | ALA3394958 | ||||||
| 2. | ALA137386 | 2a (E-isomer) | Ki | = | 1.43 | nM | ALA3394957 | 8.85 | nM | Homo sapiens | ||
| 3. | ALA137386 | 2a (E-isomer) | Ki | = | 46 | nM | ALA3394956 | 7.34 | nM | Homo sapiens | ||
| 4. | ALA137386 | 2a (E-isomer) | Ratio Ki | = | 8.1 | ALA3396877 | ||||||
| 5. | ALA137386 | 2a (E-isomer) | logP | = | 5.03 | ALA3396878 | ||||||
| 6. | ALA137386 | 2a (E-isomer) | Ki | = | 1.03 | nM | ALA3396876 | 8.99 | nM | Homo sapiens | ||
| 7. | ALA137386 | 2a (E-isomer) | Ki | = | 8.3 | nM | ALA3396875 | 8.08 | nM | Homo sapiens | ||
| 8. | ALA137386 | 2a (E-isomer) | Activity | 0 | ALA5031258 | Not Active | ||||||
| 9. | ALA137386 | 2a (E-isomer) | Activity | 0 | ALA5031257 | Active | ||||||
| 10. | ALA137386 | 2a (E-isomer) | FC | = | 43 | ALA5031254 | Homo sapiens | |||||
| 11. | ALA137386 | 2a (E-isomer) | Ki | = | 1.89 | nM | ALA5031251 | 8.72 | nM | Homo sapiens | ||
| 12. | ALA137386 | 2a (E-isomer) | Ki | = | 23.6 | nM | ALA5031250 | 7.63 | nM | Homo sapiens | ||
| 13. | ALA137386 | 2a (E-isomer) | Activity | = | 133 | % | ALA860617 | % | Mus musculus | |||
| 14. | ALA137386 | 2a (E-isomer) | Ki | = | 4.51 | nM | ALA860607 | 8.35 | nM | Homo sapiens | ||
| 15. | ALA137386 | 2a (E-isomer) | Ki | = | 103 | nM | ALA872291 | 6.99 | nM | Homo sapiens | ||
| 16. | ALA137386 | 2a (E-isomer) | Ki | = | 0.9 | nM | ALA871845 | 9.05 | nM | Homo sapiens | ||
| 17. | ALA137386 | 2a (E-isomer) | Ki | = | 3.25 | nM | ALA872399 | 8.49 | nM | Homo sapiens | ||
| 18. | ALA137386 | 2a (E-isomer) | Ki | = | 0.9 | nM | ALA876368 | 9.05 | nM | Homo sapiens | ||
| 19. | ALA137386 | 2a (E-isomer) | Ki | = | 3.25 | nM | ALA830350 | 8.49 | nM | |||
| 20. | ALA137386 | 2a (E-isomer) | Ki | = | 4.51 | nM | ALA769622 | 8.35 | nM | Homo sapiens |
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