# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4162433 | 10 | Activity | 0 | ALA4154400 | Not Active | Mus musculus | |||||
2. | ALA4162433 | 10 | ED50 | = | 10.69 | mg kg-1 | ALA4154398 | mg.kg-1 | Rattus norvegicus | |||
3. | ALA4162433 | 10 | INH | 0 | ALA4154398 | Dose-dependent effect | % | Rattus norvegicus | ||||
4. | ALA4162433 | 10 | pKb | = | 6.15 | ALA4154397 | Cavia porcellus | |||||
5. | ALA4162433 | 10 | pKb | = | 6.39 | ALA4154396 | ||||||
6. | ALA4162433 | 10 | INH | 0 | ALA4154396 | Dose-dependent effect | % | |||||
7. | ALA4162433 | 10 | INH | 0 | ALA4154395 | Dose-dependent effect | % | Cavia porcellus | ||||
8. | ALA4162433 | 10 | Activity | 0 | ALA4154394 | Not Active | ||||||
9. | ALA4162433 | 10 | Activity | 0 | ALA4154393 | Not Active | Cavia porcellus | |||||
10. | ALA4162433 | 10 | Ki | = | 37.8 | nM | ALA4154392 | 7.42 | nM | Homo sapiens | ||
11. | ALA4162433 | 10 | Drug metabolism | = | 30 | % | ALA4154404 | % | ||||
12. | ALA4162433 | 10 | Activity | 0 | ALA4154403 | Dose-dependent effect | Mus musculus | |||||
13. | ALA4162433 | 10 | Activity | 0 | ALA4154401 | Active | Mus musculus | |||||
14. | ALA4162433 | 10 | Ki | = | 37.8 | nM | ALA4734937 | 7.42 | nM | Homo sapiens |