| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4162911 | 39c | Vdss | = | 11.9 | L/Kg | ALA4137512 | L.kg-1 | Mus musculus | |||
| 2. | ALA4162911 | 39c | CL | = | 0.9 | L/hr/kg | ALA4137509 | mL.min-1.kg-1 | Mus musculus | |||
| 3. | ALA4162911 | 39c | t1/2 | = | 10.4 | hr | ALA4137506 | hr | Mus musculus | |||
| 4. | ALA4162911 | 39c | AUC | = | 8789 | nM.hr | ALA4137503 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 5. | ALA4162911 | 39c | t1/2 | = | 0.1 | hr | ALA4137500 | hr | ||||
| 6. | ALA4162911 | 39c | Stability | = | 15 | % | ALA4137499 | % | ||||
| 7. | ALA4162911 | 39c | t1/2 | > | 2.4 | hr | ALA4137498 | hr | ||||
| 8. | ALA4162911 | 39c | Stability | = | 97 | % | ALA4137497 | % | ||||
| 9. | ALA4162911 | 39c | INH | = | 4.6 | % | ALA4137496 | % | Homo sapiens | |||
| 10. | ALA4162911 | 39c | INH | = | 27.6 | % | ALA4137495 | % | Homo sapiens | |||
| 11. | ALA4162911 | 39c | INH | = | 4 | % | ALA4137494 | % | Homo sapiens | |||
| 12. | ALA4162911 | 39c | INH | = | 8 | % | ALA4137493 | % | Homo sapiens | |||
| 13. | ALA4162911 | 39c | INH | = | 28.6 | % | ALA4137492 | % | Homo sapiens | |||
| 14. | ALA4162911 | 39c | INH | > | 5 | % | ALA4137491 | % | Homo sapiens | |||
| 15. | ALA4162911 | 39c | INH | 0 | ALA4137490 | Not Active | % | Homo sapiens | ||||
| 16. | ALA4162911 | 39c | INH | = | 10 | % | ALA4137489 | % | Homo sapiens | |||
| 17. | ALA4162911 | 39c | INH | 0 | ALA4137488 | Dose-dependent effect | % | Homo sapiens | ||||
| 18. | ALA4162911 | 39c | INH | = | 0 | % | ALA4137487 | % | Mus musculus | |||
| 19. | ALA4162911 | 39c | INH | = | 81 | % | ALA4137486 | % | Homo sapiens | |||
| 20. | ALA4162911 | 39c | IC50 | > | 20 | uM | ALA4137477 | nM | Homo sapiens |
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