| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4163247 | 2; BVM | t1/2 | <= | 3 | min | ALA4157509 | hr | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | |||
| 2. | ALA4163247 | 2; BVM | t1/2 | <= | 3 | min | ALA4157508 | hr | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | |||
| 3. | ALA4163247 | 2; BVM | t1/2 | = | 51 | min | ALA4157507 | hr | Human immunodeficiency virus 1 | |||
| 4. | ALA4163247 | 2; BVM | PB | > | 99 | % | ALA4157500 | % | ||||
| 5. | ALA4163247 | 2; BVM | log(activity) | = | 0.72 | /ml | ALA4157499 | /ml | Human immunodeficiency virus 1 | |||
| 6. | ALA4163247 | 2; BVM | t1/2 | > | 120 | min | ALA4157471 | hr | ||||
| 7. | ALA4163247 | 2; BVM | t1/2 | > | 120 | min | ALA4157469 | hr | ||||
| 8. | ALA4163247 | 2; BVM | EC50 | > | 10 | uM | ALA4157406 | nM | Human immunodeficiency virus 1 | |||
| 9. | ALA4163247 | 2; BVM | solubility | < | 1 | ug ml-1 | ALA4157403 | ug.mL-1 | ||||
| 10. | ALA4163247 | 2; BVM | Kd | = | 259 | nM | ALA4157401 | 6.59 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | ||
| 11. | ALA4163247 | 2; BVM | Kd | = | 49.2 | nM | ALA4157400 | 7.31 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | ||
| 12. | ALA4163247 | 2; BVM | Kd | = | 15 | nM | ALA4157399 | 7.82 | nM | Human immunodeficiency virus type 1 group M subtype B (isolate HXB2)(HIV-1) | ||
| 13. | ALA4163247 | 2; BVM | Kd | = | 5.4 | nM | ALA4157398 | 8.27 | nM | Human immunodeficiency virus 1 | ||
| 14. | ALA4163247 | 2; BVM | EC50 | = | 77 | nM | ALA4157397 | 7.11 | nM | Human immunodeficiency virus 1 | ||
| 15. | ALA4163247 | 2; BVM | EC50 | = | 40 | nM | ALA4157396 | 7.40 | nM | Human immunodeficiency virus 1 | ||
| 16. | ALA4163247 | 2; BVM | EC50 | = | 1114 | nM | ALA4157395 | 5.95 | nM | Human immunodeficiency virus 1 | ||
| 17. | ALA4163247 | 2; BVM | EC50 | = | 1810 | nM | ALA4157394 | 5.74 | nM | Human immunodeficiency virus 1 | ||
| 18. | ALA4163247 | 2; BVM | EC50 | = | 7 | nM | ALA4157393 | 8.15 | nM | Human immunodeficiency virus 1 | ||
| 19. | ALA4163247 | 2; BVM | EC50 | = | 74 | nM | ALA4157392 | 7.13 | nM | Human immunodeficiency virus 1 | ||
| 20. | ALA4163247 | 2; BVM | AUC | = | 13743 | nM.hr | ALA4157389 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus |
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