# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4163615 | 18; M090 | INH | 0 | ALA4137000 | Dose-dependent effect | % | Influenza A virus (strain A/Aichi/2/1968 H3N2) | ||||
2. | ALA4163615 | 18; M090 | Ratio EC50 | = | 3 | ALA4137003 | Influenza A virus | |||||
3. | ALA4163615 | 18; M090 | INH | 0 | ALA4137001 | Active | % | Influenza A virus | ||||
4. | ALA4163615 | 18; M090 | IC50 | = | 1.23 | uM | ALA4137000 | 5.91 | nM | Influenza A virus (strain A/Aichi/2/1968 H3N2) | ||
5. | ALA4163615 | 18; M090 | INH | 0 | ALA4136999 | Dose-dependent effect | % | Influenza A virus (A/Puerto Rico/8/1934(H1N1)) | ||||
6. | ALA4163615 | 18; M090 | EC50 | > | 43 | uM | ALA4136998 | nM | Influenza A virus | |||
7. | ALA4163615 | 18; M090 | EC50 | > | 43 | uM | ALA4136997 | nM | Influenza A virus | |||
8. | ALA4163615 | 18; M090 | EC50 | > | 43 | uM | ALA4136996 | nM | Influenza A virus | |||
9. | ALA4163615 | 18; M090 | EC50 | = | 25.6 | uM | ALA4136995 | 4.59 | nM | Influenza A virus | ||
10. | ALA4163615 | 18; M090 | EC50 | = | 13.8 | uM | ALA4136994 | 4.86 | nM | Influenza A virus | ||
11. | ALA4163615 | 18; M090 | EC50 | = | 8.7 | uM | ALA4136993 | 5.06 | nM | Influenza A virus | ||
12. | ALA4163615 | 18; M090 | EC50 | = | 1.7 | uM | ALA4136992 | 5.77 | nM | Influenza A virus | ||
13. | ALA4163615 | 18; M090 | EC50 | = | 0.32 | uM | ALA4136991 | 6.50 | nM | Influenza A virus | ||
14. | ALA4163615 | 18; M090 | EC50 | = | 0.34 | uM | ALA4136990 | 6.47 | nM | Influenza A virus | ||
15. | ALA4163615 | 18; M090 | INH | 0 | ALA4136989 | Not Active | % | Influenza A virus (A/Puerto Rico/8/1934(H1N1)) | ||||
16. | ALA4163615 | 18; M090 | INH | 0 | ALA4136988 | Not Active | % | Influenza A virus (A/Udorn/307/1972(H3N2)) | ||||
17. | ALA4163615 | 18; M090 | INH | 0 | ALA4136987 | Active | % | Influenza A virus | ||||
18. | ALA4163615 | 18; M090 | EC50 | = | 0.1 | uM | ALA4136986 | 7.00 | nM | Influenza A virus | ||
19. | ALA4163615 | 18; M090 | EC50 | = | 0.34 | uM | ALA4136985 | 6.47 | nM | Influenza A virus | ||
20. | ALA4163615 | 18; M090 | EC50 | = | 6.79 | uM | ALA4136984 | 5.17 | nM | Influenza A virus |