| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4165147 | AP5 | EC50 | > | 10 | uM | ALA4151317 | nM | Homo sapiens | |||
| 2. | ALA4165147 | AP5 | logD | = | 2.51 | ALA4151316 | ||||||
| 3. | ALA4165147 | AP5 | Activity | 0 | ALA4151315 | Non-Toxic | Rattus norvegicus | |||||
| 4. | ALA4165147 | AP5 | Activity | 0 | ALA4151314 | Non-Toxic | Rattus norvegicus | |||||
| 5. | ALA4165147 | AP5 | Activity | 0 | ALA4151313 | Non-Toxic | Rattus norvegicus | |||||
| 6. | ALA4165147 | AP5 | Activity | 0 | ALA4151312 | Non-Toxic | Rattus norvegicus | |||||
| 7. | ALA4165147 | AP5 | Activity | 0 | ALA4151311 | Non-Toxic | Rattus norvegicus | |||||
| 8. | ALA4165147 | AP5 | Activity | = | 90 | % | ALA4151310 | % | Rattus norvegicus | |||
| 9. | ALA4165147 | AP5 | Tmax | = | 1 | hr | ALA4151309 | hr | Rattus norvegicus | |||
| 10. | ALA4165147 | AP5 | Cmin | = | 328 | uM | ALA4151308 | uM | Rattus norvegicus | |||
| 11. | ALA4165147 | AP5 | Cmax | = | 545 | uM | ALA4151307 | nM | Rattus norvegicus | |||
| 12. | ALA4165147 | AP5 | AUC | = | 7354 | uM.hr | ALA4151306 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 13. | ALA4165147 | AP5 | Activity | = | 72 | % | ALA4151305 | % | Rattus norvegicus | |||
| 14. | ALA4165147 | AP5 | Tmax | = | 1 | hr | ALA4151304 | hr | Rattus norvegicus | |||
| 15. | ALA4165147 | AP5 | Cmin | = | 70 | uM | ALA4151303 | uM | Rattus norvegicus | |||
| 16. | ALA4165147 | AP5 | Cmax | = | 223 | uM | ALA4151302 | nM | Rattus norvegicus | |||
| 17. | ALA4165147 | AP5 | AUC | = | 2309 | uM.hr | ALA4151301 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Rattus norvegicus | ||
| 18. | ALA4165147 | AP5 | Drug metabolism | = | 75 | % | ALA4151298 | % | ||||
| 19. | ALA4165147 | AP5 | Drug metabolism | 0 | ALA4151297 | Metabolite_Notdetected | ||||||
| 20. | ALA4165147 | AP5 | CLH | = | 102 | ml/min.kg | ALA4151296 | mL.min-1.kg-1 |
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