| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4165748 | 12 | INH | = | 19 | % | ALA4158290 | % | Mus musculus | |||
| 2. | ALA4165748 | 12 | fAUC/dose | = | 4.7 | uM.min | ALA4158288 | uM.min | Mus musculus | |||
| 3. | ALA4165748 | 12 | fAUC/dose | = | 2.1 | uM.min | ALA4158287 | uM.min | Rattus norvegicus | |||
| 4. | ALA4165748 | 12 | F | = | 35 | % | ALA4158286 | % | Rattus norvegicus | |||
| 5. | ALA4165748 | 12 | t1/2 | = | 431 | min | ALA4158285 | hr | Rattus norvegicus | |||
| 6. | ALA4165748 | 12 | CL free | = | 342 | ml/min.kg | ALA4158284 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 7. | ALA4165748 | 12 | Fu | = | 0.011 | ALA4158283 | ||||||
| 8. | ALA4165748 | 12 | Fu | = | 0.007 | ALA4158282 | ||||||
| 9. | ALA4165748 | 12 | logD | = | 2.2 | ALA4158275 | ||||||
| 10. | ALA4165748 | 12 | pEC50 | = | 7.6 | ALA4158276 | 7.60 | nM | Homo sapiens | |||
| 11. | ALA4165748 | 12 | pEC50 | = | 6.9 | ALA4158277 | 6.90 | nM | Mus musculus | |||
| 12. | ALA4165748 | 12 | Emax | = | 103 | % | ALA4158278 | % | Homo sapiens | |||
| 13. | ALA4165748 | 12 | Emax | = | 84 | % | ALA4158279 | % | Mus musculus | |||
| 14. | ALA4165748 | 12 | pKi | = | 6.6 | ALA4158280 | 6.60 | nM | Homo sapiens |
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