# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4168827 | 6b | INH | 0 | ALA4149796 | Dose-dependent effect | % | Homo sapiens | ||||
2. | ALA4168827 | 6b | INH | = | 41 | % | ALA4149795 | % | Homo sapiens | |||
3. | ALA4168827 | 6b | Ki | = | 0.53 | uM | ALA4149762 | 6.28 | nM | Homo sapiens | ||
4. | ALA4168827 | 6b | solubility | = | 56 | uM | ALA4149760 | nM | ||||
5. | ALA4168827 | 6b | Papp | = | 11 | 10'-6 cm/s | ALA4149759 | 10'-6 cm/s | ||||
6. | ALA4168827 | 6b | CLH(app) | > | 560 | microL/min/mg | ALA4149758 | mL.min-1.g-1 | ||||
7. | ALA4168827 | 6b | logD | = | 3 | ALA4149757 | ||||||
8. | ALA4168827 | 6b | IC50 | > | 60 | uM | ALA4149756 | nM | Homo sapiens | |||
9. | ALA4168827 | 6b | IC50 | > | 26 | uM | ALA4149755 | nM | Homo sapiens | |||
10. | ALA4168827 | 6b | IC50 | > | 60 | uM | ALA4149754 | nM | Homo sapiens | |||
11. | ALA4168827 | 6b | IC50 | > | 60 | uM | ALA4149753 | nM | Homo sapiens | |||
12. | ALA4168827 | 6b | IC50 | > | 60 | uM | ALA4149752 | nM | Homo sapiens | |||
13. | ALA4168827 | 6b | IC50 | = | 0.12 | uM | ALA4149751 | 6.92 | nM | Homo sapiens |