# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4172741 | 39 | Stabilty | = | 74 | % | ALA4714701 | % | ||||
2. | ALA4172741 | 39 | IC50 | = | 4.4 | uM | ALA4714699 | 5.36 | nM | |||
3. | ALA4172741 | 39 | Activity | = | 93.6 | % | ALA4714698 | % | ||||
4. | ALA4172741 | 39 | Activity | = | 17.5 | % | ALA4714697 | % | ||||
5. | ALA4172741 | 39 | t1/2 | = | 1.3 | hr | ALA4678392 | hr | ||||
6. | ALA4172741 | 39 | Drug metabolism | 0 | ALA4158747 | Metabolite_Detected | ||||||
7. | ALA4172741 | 39 | Activity | 0 | ALA4158746 | Non-Toxic | Mus musculus | |||||
8. | ALA4172741 | 39 | Drug metabolism | 0 | ALA4158745 | Metabolite_Notdetected | ||||||
9. | ALA4172741 | 39 | Activity | 0 | ALA4158716 | Active | Mus musculus | |||||
10. | ALA4172741 | 39 | Activity | 0 | ALA4158715 | Active | Mus musculus | |||||
11. | ALA4172741 | 39 | Activity | 0 | ALA4158714 | Active | Mus musculus | |||||
12. | ALA4172741 | 39 | Cp | = | 1.2 | uM | ALA4158713 | uM | ||||
13. | ALA4172741 | 39 | Vd | = | 32 | L/Kg | ALA4158711 | L.kg-1 | Mus musculus | |||
14. | ALA4172741 | 39 | CL | = | 17 | L/hr/kg | ALA4158709 | mL.min-1.kg-1 | Mus musculus | |||
15. | ALA4172741 | 39 | Cmax | = | 640 | ug/L | ALA4158712 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
16. | ALA4172741 | 39 | t1/2 | = | 1.3 | hr | ALA4158710 | hr | Mus musculus | |||
17. | ALA4172741 | 39 | Activity | 0 | ALA4158708 | Non-Toxic | Mus musculus | |||||
18. | ALA4172741 | 39 | Activity | 0 | ALA4158707 | Non-Toxic | Mus musculus | |||||
19. | ALA4172741 | 39 | Activity | 0 | ALA4158706 | Non-Toxic | Mus musculus | |||||
20. | ALA4172741 | 39 | Activity | 0 | ALA4158705 | Non-Toxic | Mus musculus |