| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4172928 | 3 | INH | = | 5 | % | ALA4158290 | % | Mus musculus | |||
| 2. | ALA4172928 | 3 | fAUC/dose | = | 0.32 | uM.min | ALA4158288 | uM.min | Mus musculus | |||
| 3. | ALA4172928 | 3 | fAUC/dose | = | 0.26 | uM.min | ALA4158287 | uM.min | Rattus norvegicus | |||
| 4. | ALA4172928 | 3 | F | = | 47 | % | ALA4158286 | % | Rattus norvegicus | |||
| 5. | ALA4172928 | 3 | t1/2 | = | 590 | min | ALA4158285 | hr | Rattus norvegicus | |||
| 6. | ALA4172928 | 3 | CL free | = | 2800 | ml/min.kg | ALA4158284 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 7. | ALA4172928 | 3 | Fu | = | 0 | ALA4158283 | ||||||
| 8. | ALA4172928 | 3 | Fu | = | 0 | ALA4158282 | ||||||
| 9. | ALA4172928 | 3 | logD | = | 3 | ALA4158275 | ||||||
| 10. | ALA4172928 | 3 | pEC50 | = | 7.9 | ALA4158276 | 7.90 | nM | Homo sapiens | |||
| 11. | ALA4172928 | 3 | pEC50 | = | 7.3 | ALA4158277 | 7.30 | nM | Mus musculus | |||
| 12. | ALA4172928 | 3 | Emax | = | 125 | % | ALA4158278 | % | Homo sapiens | |||
| 13. | ALA4172928 | 3 | Emax | = | 113 | % | ALA4158279 | % | Mus musculus | |||
| 14. | ALA4172928 | 3 | pKi | = | 6.7 | ALA4158280 | 6.70 | nM | Homo sapiens | |||
| 15. | ALA4172928 | 3 | pEC50 | = | 6.68 | ALA4158156 | 6.68 | nM | Homo sapiens | |||
| 16. | ALA4172928 | 3 | EC50 | = | 14 | nM | ALA4669442 | 7.85 | nM | Homo sapiens |
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