| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4173663 | 11 | INH | = | 40 | % | ALA4158290 | % | Mus musculus | |||
| 2. | ALA4173663 | 11 | fAUC/dose | = | 0.53 | uM.min | ALA4158288 | uM.min | Mus musculus | |||
| 3. | ALA4173663 | 11 | fAUC/dose | = | 0.07 | uM.min | ALA4158287 | uM.min | Rattus norvegicus | |||
| 4. | ALA4173663 | 11 | F | = | 25 | % | ALA4158286 | % | Rattus norvegicus | |||
| 5. | ALA4173663 | 11 | t1/2 | = | 155 | min | ALA4158285 | hr | Rattus norvegicus | |||
| 6. | ALA4173663 | 11 | CL free | = | 6692 | ml/min.kg | ALA4158284 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 7. | ALA4173663 | 11 | Fu | = | 0.001 | ALA4158283 | ||||||
| 8. | ALA4173663 | 11 | Fu | = | 0.001 | ALA4158282 | ||||||
| 9. | ALA4173663 | 11 | logD | = | 3.1 | ALA4158275 | ||||||
| 10. | ALA4173663 | 11 | pEC50 | = | 7.6 | ALA4158276 | 7.60 | nM | Homo sapiens | |||
| 11. | ALA4173663 | 11 | pEC50 | = | 7.1 | ALA4158277 | 7.10 | nM | Mus musculus | |||
| 12. | ALA4173663 | 11 | Emax | = | 108 | % | ALA4158278 | % | Homo sapiens | |||
| 13. | ALA4173663 | 11 | Emax | = | 72 | % | ALA4158279 | % | Mus musculus | |||
| 14. | ALA4173663 | 11 | pKi | = | 7.2 | ALA4158280 | 7.20 | nM | Homo sapiens |
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