# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4174219 | 58 | Activity | = | 60 | % | ALA5152584 | % | ||||
2. | ALA4174219 | 58 | Activity | = | 100 | % | ALA5152583 | % | ||||
3. | ALA4174219 | 58 | IC90 | = | 0.77 | uM | ALA5152581 | nM | Homo sapiens | |||
4. | ALA4174219 | 58 | PPB | = | 99.8 | % | ALA5152580 | % | ||||
5. | ALA4174219 | 58 | beta t1/2 | = | 2.4 | hr | ALA5152579 | hr | ||||
6. | ALA4174219 | 58 | AUC | = | 415 | umol/l.hr | ALA4130828 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
7. | ALA4174219 | 58 | Cmax | = | 105 | umol/L | ALA4130827 | nM | Mus musculus | |||
8. | ALA4174219 | 58 | t1/2 | = | 2.5 | hr | ALA4130826 | hr | Mus musculus | |||
9. | ALA4174219 | 58 | Activity | = | 98.7 | % | ALA4130820 | % | ||||
10. | ALA4174219 | 58 | INH | = | 95.6 | % | ALA4130819 | % | Homo sapiens | |||
11. | ALA4174219 | 58 | IC50 | = | 6.65 | uM | ALA4130818 | 5.18 | nM | Homo sapiens |