| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4174883 | 20b | CLH | = | 8.6 | microL/min/mg | ALA4146174 | mL.min-1.g-1 | ||||
| 2. | ALA4174883 | 20b | CLH | = | 27.8 | microL/min/mg | ALA4146173 | mL.min-1.g-1 | ||||
| 3. | ALA4174883 | 20b | t1/2 | = | 270.7 | min | ALA4146172 | hr | ||||
| 4. | ALA4174883 | 20b | t1/2 | = | 83.2 | min | ALA4146171 | hr | ||||
| 5. | ALA4174883 | 20b | solubility | > | 100 | uM | ALA4146170 | nM | ||||
| 6. | ALA4174883 | 20b | Ratio | = | 25 | ALA4146169 | Mycobacterium tuberculosis | |||||
| 7. | ALA4174883 | 20b | Ratio IC50 | = | 8.95 | ALA4146168 | ||||||
| 8. | ALA4174883 | 20b | IC50 | = | 11.99 | uM | ALA4146167 | 4.92 | nM | Homo sapiens | ||
| 9. | ALA4174883 | 20b | IC50 | = | 1.34 | uM | ALA4146166 | 5.87 | nM | Mycobacterium tuberculosis | ||
| 10. | ALA4174883 | 20b | Selectivity Index | > | 4000 | ALA4146165 | ||||||
| 11. | ALA4174883 | 20b | LC50 | > | 100 | uM | ALA4146164 | nM | ||||
| 12. | ALA4174883 | 20b | CC50 | > | 100 | uM | ALA4146163 | nM | Homo sapiens | |||
| 13. | ALA4174883 | 20b | MIC90 | = | 0.025 | uM | ALA4146162 | nM | Mycobacterium tuberculosis | |||
| 14. | ALA4174883 | 20b | MIC50 | = | 0.01 | uM | ALA4146162 | nM | Mycobacterium tuberculosis | |||
| 15. | ALA4174883 | 20b | MIC90 | = | 0.2 | uM | ALA4146161 | nM | Mycobacterium tuberculosis | |||
| 16. | ALA4174883 | 20b | MIC50 | = | 0.02 | uM | ALA4146161 | nM | Mycobacterium tuberculosis | |||
| 17. | ALA4174883 | 20b | Activity | = | 88.4 | % | ALA4146160 | % | Mycobacterium tuberculosis |
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