# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4176183 | 52 | IC50 | = | 14.9 | nM | ALA4158231 | 7.83 | nM | Homo sapiens | ||
2. | ALA4176183 | 52 | INH | > | 90 | % | ALA4158230 | % | Homo sapiens | |||
3. | ALA4176183 | 52 | Ratio IC50 | <= | 5 | ALA4158227 | ||||||
4. | ALA4176183 | 52 | Ratio IC50 | <= | 5 | ALA4158226 | ||||||
5. | ALA4176183 | 52 | Ratio IC50 | <= | 5 | ALA4158225 | ||||||
6. | ALA4176183 | 52 | Ratio IC50 | <= | 5 | ALA4158224 | Homo sapiens | |||||
7. | ALA4176183 | 52 | Ratio IC50 | <= | 5 | ALA4158223 | Homo sapiens | |||||
8. | ALA4176183 | 52 | IC50 | > | 5 | uM | ALA4158222 | nM | Homo sapiens | |||
9. | ALA4176183 | 52 | IC50 | > | 5 | uM | ALA4158221 | nM | Homo sapiens | |||
10. | ALA4176183 | 52 | IC50 | = | 1100 | nM | ALA4158220 | 5.96 | nM | Homo sapiens | ||
11. | ALA4176183 | 52 | IC50 | > | 5000 | nM | ALA4158219 | nM | Homo sapiens | |||
12. | ALA4176183 | 52 | IC50 | > | 5 | uM | ALA4158218 | nM | Homo sapiens | |||
13. | ALA4176183 | 52 | IC50 | = | 7.1 | nM | ALA4158215 | 8.15 | nM | Homo sapiens | ||
14. | ALA4176183 | 52 | R% | = | 40 | % | ALA4158214 | % | ||||
15. | ALA4176183 | 52 | t1/2 | = | 26 | min | ALA4158213 | hr | ||||
16. | ALA4176183 | 52 | t1/2 | = | 9 | min | ALA4158212 | hr | ||||
17. | ALA4176183 | 52 | Kinetic_solubility | 0 | ALA4158209 | Not Determined | ||||||
18. | ALA4176183 | 52 | permeability | = | 34.3 | nm/s | ALA4158210 | nm/s | ||||
19. | ALA4176183 | 52 | t1/2 | = | 12 | min | ALA4158211 | hr |