| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4177037 | 13 | INH | = | 26 | % | ALA4158290 | % | Mus musculus | |||
| 2. | ALA4177037 | 13 | fAUC/dose | = | 3.3 | uM.min | ALA4158288 | uM.min | Mus musculus | |||
| 3. | ALA4177037 | 13 | fAUC/dose | = | 0.55 | uM.min | ALA4158287 | uM.min | Rattus norvegicus | |||
| 4. | ALA4177037 | 13 | F | = | 29 | % | ALA4158286 | % | Rattus norvegicus | |||
| 5. | ALA4177037 | 13 | t1/2 | = | 280 | min | ALA4158285 | hr | Rattus norvegicus | |||
| 6. | ALA4177037 | 13 | CL free | = | 1091 | ml/min.kg | ALA4158284 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 7. | ALA4177037 | 13 | Fu | = | 0.008 | ALA4158283 | ||||||
| 8. | ALA4177037 | 13 | Fu | = | 0.006 | ALA4158282 | ||||||
| 9. | ALA4177037 | 13 | logD | = | 2.4 | ALA4158275 | ||||||
| 10. | ALA4177037 | 13 | pEC50 | = | 7.6 | ALA4158276 | 7.60 | nM | Homo sapiens | |||
| 11. | ALA4177037 | 13 | pEC50 | = | 7 | ALA4158277 | 7.00 | nM | Mus musculus | |||
| 12. | ALA4177037 | 13 | Emax | = | 104 | % | ALA4158278 | % | Homo sapiens | |||
| 13. | ALA4177037 | 13 | Emax | = | 88 | % | ALA4158279 | % | Mus musculus | |||
| 14. | ALA4177037 | 13 | pKi | = | 6.8 | ALA4158280 | 6.80 | nM | Homo sapiens |
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