| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4202712 | 10k | Activity | 0 | ALA4198067 | Not Active | Homo sapiens | |||||
| 2. | ALA4202712 | 10k | Activity | 0 | ALA4198066 | Not Active | Homo sapiens | |||||
| 3. | ALA4202712 | 10k | Activity | 0 | ALA4198065 | Not Active | Homo sapiens | |||||
| 4. | ALA4202712 | 10k | Activity | 0 | ALA4198064 | Dose-dependent effect | Homo sapiens | |||||
| 5. | ALA4202712 | 10k | CLH | = | 5.9 | ml/min.kg | ALA4198063 | mL.min-1.kg-1 | ||||
| 6. | ALA4202712 | 10k | t1/2 | = | 3.5 | hr | ALA4198062 | hr | ||||
| 7. | ALA4202712 | 10k | CLH | = | 29 | ml/min.kg | ALA4198061 | mL.min-1.kg-1 | ||||
| 8. | ALA4202712 | 10k | t1/2 | = | 1.62 | hr | ALA4198060 | hr | ||||
| 9. | ALA4202712 | 10k | CLH | = | 47.8 | ml/min.kg | ALA4198059 | mL.min-1.kg-1 | ||||
| 10. | ALA4202712 | 10k | t1/2 | = | 1.2 | hr | ALA4198058 | hr | ||||
| 11. | ALA4202712 | 10k | Ratio IC50 | = | 0.21 | ALA4198057 | ||||||
| 12. | ALA4202712 | 10k | Ratio IC50 | = | 0.15 | ALA4198056 | ||||||
| 13. | ALA4202712 | 10k | IC50 | = | 0.05 | uM | ALA4198055 | 7.30 | nM | Homo sapiens | ||
| 14. | ALA4202712 | 10k | IC50 | = | 0.24 | uM | ALA4198054 | 6.62 | nM | Homo sapiens | ||
| 15. | ALA4202712 | 10k | IC50 | = | 0.25 | uM | ALA4198053 | 6.60 | nM | |||
| 16. | ALA4202712 | 10k | IC50 | = | 1.71 | uM | ALA4198052 | 5.77 | nM | Homo sapiens | ||
| 17. | ALA4202712 | 10k | Ratio IC50 | = | 4.8 | ALA4198051 | ||||||
| 18. | ALA4202712 | 10k | IC50 | = | 3.8 | uM | ALA4198050 | 5.42 | nM | |||
| 19. | ALA4202712 | 10k | IC50 | = | 0.8 | uM | ALA4198049 | 6.10 | nM | Homo sapiens | ||
| 20. | ALA4202712 | 10k | IC50 | = | 7.7 | uM | ALA4198048 | 5.11 | nM | Homo sapiens |
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