| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4206372 | 9 | INH | 0 | ALA4704020 | Not Determined | % | Homo sapiens | ||||
| 2. | ALA4206372 | 9 | IC50 | = | 2.4 | uM | ALA4704019 | 5.62 | nM | Homo sapiens | ||
| 3. | ALA4206372 | 9 | IC50 | = | 4170 | nM | ALA4704018 | 5.38 | nM | Mus musculus | ||
| 4. | ALA4206372 | 9 | IC50 | = | 84 | nM | ALA4704017 | 7.08 | nM | Homo sapiens | ||
| 5. | ALA4206372 | 9 | IC50 | = | 29 | nM | ALA4704015 | 7.54 | nM | Mus musculus | ||
| 6. | ALA4206372 | 9 | IC50 | = | 1250 | nM | ALA4704014 | 5.90 | nM | Homo sapiens | ||
| 7. | ALA4206372 | 9 | Ratio IC50 | = | 143 | ALA4184960 | ||||||
| 8. | ALA4206372 | 9 | AUC | = | 1.75 | mg.hr/L | ALA4184961 | ng.hr.mL-1 | Mus musculus | |||
| 9. | ALA4206372 | 9 | Cmax | = | 1.48 | mg/L | ALA4184962 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 10. | ALA4206372 | 9 | CL | = | 1.71 | L/hr/kg | ALA4184963 | mL.min-1.kg-1 | Mus musculus | |||
| 11. | ALA4206372 | 9 | Vdss | = | 4.6 | L/Kg | ALA4184964 | L.kg-1 | Mus musculus | |||
| 12. | ALA4206372 | 9 | t1/2 | = | 2.87 | hr | ALA4184965 | hr | Mus musculus | |||
| 13. | ALA4206372 | 9 | AUC | = | 3.57 | mg.hr/L | ALA4184966 | ng.hr.mL-1 | Mus musculus | |||
| 14. | ALA4206372 | 9 | Cmax | = | 0.84 | mg/L | ALA4184967 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Mus musculus | ||
| 15. | ALA4206372 | 9 | Tmax | = | 0.5 | hr | ALA4184968 | hr | Mus musculus | |||
| 16. | ALA4206372 | 9 | t1/2 | = | 2.83 | hr | ALA4184969 | hr | Mus musculus | |||
| 17. | ALA4206372 | 9 | F | = | 61.2 | % | ALA4184970 | % | Mus musculus | |||
| 18. | ALA4206372 | 9 | IC50 | = | 29 | nM | ALA4184958 | 7.54 | nM | Mus musculus | ||
| 19. | ALA4206372 | 9 | IC50 | = | 4170 | nM | ALA4184959 | 5.38 | nM | Mus musculus |
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