# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4206601 | 3 | Km | = | 0.081 | nM | ALA4180659 | nM | Rattus norvegicus | |||
2. | ALA4206601 | 3 | Vmax | = | 6.019 | 10'4OD/sec | ALA4180658 | 10'4OD/sec | Rattus norvegicus | |||
3. | ALA4206601 | 3 | pIC50 | = | 7.9 | ALA4180641 | 7.90 | nM | Rattus norvegicus | |||
4. | ALA4206601 | 3 | INH | 0 | ALA4180657 | Dose-dependent effect | % | Rattus norvegicus | ||||
5. | ALA4206601 | 3 | Activity | = | 249.3 | nmol/g | ALA4180655 | nmol/g | Rattus norvegicus | |||
6. | ALA4206601 | 3 | Activity | = | 375.3 | nmol/g | ALA4180654 | nmol/g | Rattus norvegicus | |||
7. | ALA4206601 | 3 | Activity | = | 440.1 | nmol/g | ALA4180653 | nmol/g | Rattus norvegicus | |||
8. | ALA4206601 | 3 | Activity | = | 656.7 | nmol/g | ALA4180652 | nmol/g | Rattus norvegicus | |||
9. | ALA4206601 | 3 | Ki | = | 66.1 | nM | ALA4180651 | 7.18 | nM | Homo sapiens | ||
10. | ALA4206601 | 3 | Ki | = | 16.9 | nM | ALA4180650 | 7.77 | nM | Rattus norvegicus | ||
11. | ALA4206601 | 3 | Vmax | = | 0.063 | 10'4OD/sec | ALA4180649 | 10'4OD/sec | Homo sapiens | |||
12. | ALA4206601 | 3 | Km | = | 0.036 | mmol/L | ALA4180648 | nM | Homo sapiens | |||
13. | ALA4206601 | 3 | IC50 | = | 83.5 | nM | ALA4180647 | 7.08 | nM | Homo sapiens | ||
14. | ALA4206601 | 3 | IC50 | = | 9434 | nM | ALA4180646 | 5.03 | nM | Homo sapiens | ||
15. | ALA4206601 | 3 | Ratio IC50 | = | 792 | ALA4180645 | ||||||
16. | ALA4206601 | 3 | Km | = | 0.101 | nM | ALA4180644 | nM | Rattus norvegicus | |||
17. | ALA4206601 | 3 | Vmax | = | 7.154 | 10'4OD/sec | ALA4180643 | 10'4OD/sec | Rattus norvegicus | |||
18. | ALA4206601 | 3 | IC50 | = | 9.98 | uM | ALA4180642 | 5.00 | nM | Rattus norvegicus | ||
19. | ALA4206601 | 3 | IC50 | = | 12.6 | nM | ALA4180641 | 7.90 | nM | Rattus norvegicus | ||
20. | ALA4206601 | 3 | Km | = | 0.022 | mmol/L | ALA4180660 | nM | Homo sapiens |