# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | [³H]TBZOH | [3H]-DHTB | Bmax | = | 41.2 | pmol/mg | ALA4202143 | pmol/mg | Homo sapiens | |||
2. | [³H]TBZOH | [3H]-DHTB | Activity | 0 | ALA4202138 | Active | Homo sapiens | |||||
3. | [³H]TBZOH | [3H]-DHTB | Activity | 0 | ALA4202152 | Non-Toxic | Homo sapiens | |||||
4. | [³H]TBZOH | [3H]-DHTB | Ki | = | 6.7 | nM | ALA4202147 | 8.17 | nM | Homo sapiens | ||
5. | [³H]TBZOH | [3H]-DHTB | IC50 | = | 19.8 | nM | ALA4202146 | 7.70 | nM | Mus musculus | ||
6. | [³H]TBZOH | [3H]-DHTB | IC50 | = | 28.1 | nM | ALA4202145 | 7.55 | nM | Homo sapiens | ||
7. | [³H]TBZOH | [3H]-DHTB | Ki | > | 10 | uM | ALA4202144 | nM | Homo sapiens | |||
8. | [³H]TBZOH | [3H]-DHTB | Kd | = | 71 | nM | ALA4202143 | 7.15 | nM | Homo sapiens | ||
9. | [³H]TBZOH | [3H]-DHTB | Ki | = | 70 | nM | ALA4202137 | 7.16 | nM | Homo sapiens | ||
10. | [³H]TBZOH | [3H]-DHTB | Ki | = | 152 | nM | ALA4202136 | 6.82 | nM | Homo sapiens |