| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4207216 | 6a | IC50 | = | 41 | nM | ALA4199684 | 7.39 | nM | Homo sapiens | ||
| 2. | ALA4207216 | 6a | IC50 | = | 76 | nM | ALA4199685 | 7.12 | nM | Homo sapiens | ||
| 3. | ALA4207216 | 6a | IC50 | > | 37000 | nM | ALA4199686 | nM | Homo sapiens | |||
| 4. | ALA4207216 | 6a | pKa | = | 4.8 | ALA4199688 | ||||||
| 5. | ALA4207216 | 6a | Cmax | = | 32 | uM | ALA4199689 | nM | Mus musculus | |||
| 6. | ALA4207216 | 6a | AUC | = | 24 | uM.hr | ALA4199690 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 7. | ALA4207216 | 6a | CL | = | 2.1 | ml/min.kg | ALA4199691 | mL.min-1.kg-1 | Mus musculus | |||
| 8. | ALA4207216 | 6a | t1/2 | = | 3.4 | hr | ALA4199692 | hr | Mus musculus | |||
| 9. | ALA4207216 | 6a | Cmax | = | 8.2 | uM | ALA4199693 | nM | Mus musculus | |||
| 10. | ALA4207216 | 6a | AUC | = | 18 | uM.hr | ALA4199694 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 11. | ALA4207216 | 6a | t1/2 | = | 3.2 | hr | ALA4199695 | hr | Mus musculus | |||
| 12. | ALA4207216 | 6a | F | = | 76 | % | ALA4199696 | % | Mus musculus | |||
| 13. | ALA4207216 | 6a | IC50 | = | 1760 | nM | ALA4199697 | 5.75 | nM | Homo sapiens | ||
| 14. | ALA4207216 | 6a | Ratio IC50 | = | 11 | ALA4199698 | Homo sapiens |
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