| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4208344 | 17b | PB | > | 99 | % | ALA4189902 | % | ||||
| 2. | ALA4208344 | 17b | Activity | < | 10 | % | ALA4189894 | % | Homo sapiens | |||
| 3. | ALA4208344 | 17b | Activity | < | 10 | % | ALA4189893 | % | Homo sapiens | |||
| 4. | ALA4208344 | 17b | Activity | < | 10 | % | ALA4189892 | % | Homo sapiens | |||
| 5. | ALA4208344 | 17b | LD50 | > | 25 | uM | ALA4189891 | uM | Homo sapiens | |||
| 6. | ALA4208344 | 17b | Activity | = | 9 | % | ALA4189890 | % | Homo sapiens | |||
| 7. | ALA4208344 | 17b | MIC | = | 1.4 | uM | ALA4189881 | nM | Mycobacterium tuberculosis | |||
| 8. | ALA4208344 | 17b | MIC | = | 1 | uM | ALA4189880 | nM | Mycobacterium tuberculosis | |||
| 9. | ALA4208344 | 17b | MIC | = | 6 | uM | ALA4189879 | nM | Mycobacterium tuberculosis | |||
| 10. | ALA4208344 | 17b | MIC | = | 2 | uM | ALA4189878 | nM | Mycobacterium tuberculosis | |||
| 11. | ALA4208344 | 17b | beta t1/2 | = | 5 | hr | ALA4189901 | hr | Mus musculus | |||
| 12. | ALA4208344 | 17b | Tmax | = | 0.5 | hr | ALA4189900 | hr | Mus musculus | |||
| 13. | ALA4208344 | 17b | Cmax | = | 3 | uM | ALA4189899 | nM | Mus musculus | |||
| 14. | ALA4208344 | 17b | Drug metabolism | 0 | ALA4189898 | Metabolite_Notdetected | ||||||
| 15. | ALA4208344 | 17b | t1/2 | = | 26 | min | ALA4189897 | hr | ||||
| 16. | ALA4208344 | 17b | Selectivity Index | > | 10 | ALA4189895 | ||||||
| 17. | ALA4208344 | 17b | Ratio Ki(app) | = | 60 | ALA4189889 | ||||||
| 18. | ALA4208344 | 17b | Ki(app) | = | 1.1 | uM | ALA4189886 | 5.96 | nM | Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) | ||
| 19. | ALA4208344 | 17b | MIC | > | 100 | uM | ALA4189885 | nM | Mycobacterium tuberculosis | |||
| 20. | ALA4208344 | 17b | MIC | = | 3.1 | uM | ALA4189884 | nM | Mycobacterium tuberculosis |
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