# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4208555 | 39 | Drug uptake | = | 640 | ug/g | ALA4190666 | ug/g | ||||
2. | ALA4208555 | 39 | Drug uptake | = | 3128 | ug/g | ALA4190665 | ug/g | ||||
3. | ALA4208555 | 39 | permeability | = | 0.1 | 10'-5cm/hr | ALA4190664 | 10'-5cm/hr | ||||
4. | ALA4208555 | 39 | F | = | 5 | % | ALA4190663 | % | Rattus norvegicus | |||
5. | ALA4208555 | 39 | t1/2 | = | 4.4 | hr | ALA4190662 | hr | Rattus norvegicus | |||
6. | ALA4208555 | 39 | Vdss | = | 3.99 | L/Kg | ALA4190661 | L.kg-1 | Rattus norvegicus | |||
7. | ALA4208555 | 39 | CL | = | 42 | ml/min.kg | ALA4190660 | mL.min-1.kg-1 | Rattus norvegicus | |||
8. | ALA4208555 | 39 | IC50 | = | 0.72 | nM | ALA4190659 | 9.14 | nM | Homo sapiens | ||
9. | ALA4208555 | 39 | IC50 | >= | 3000 | nM | ALA4190658 | nM | ||||
10. | ALA4208555 | 39 | IC50 | = | 20 | nM | ALA4190657 | 7.70 | nM | |||
11. | ALA4208555 | 39 | IC50 | = | 450 | nM | ALA4190656 | 6.35 | nM | Homo sapiens | ||
12. | ALA4208555 | 39 | IC50 | = | 2164 | nM | ALA4190655 | 5.67 | nM | Homo sapiens | ||
13. | ALA4208555 | 39 | IC50 | = | 11405 | nM | ALA4190654 | 4.94 | nM | Homo sapiens | ||
14. | ALA4208555 | 39 | IC50 | = | 11781 | nM | ALA4190653 | 4.93 | nM | Homo sapiens | ||
15. | ALA4208555 | 39 | IC50 | = | 3152 | nM | ALA4190652 | 5.50 | nM | Homo sapiens | ||
16. | ALA4208555 | 39 | IC50 | > | 30000 | nM | ALA4190651 | nM | Homo sapiens | |||
17. | ALA4208555 | 39 | IC50 | = | 730 | nM | ALA4190650 | 6.14 | nM | |||
18. | ALA4208555 | 39 | IC50 | = | 2.3 | uM | ALA4190620 | 5.64 | nM | |||
19. | ALA4208555 | 39 | Ki | = | 25700 | nM | ALA4190649 | 4.59 | nM | Homo sapiens | ||
20. | ALA4208555 | 39 | INH | > | 3000 | nM | ALA4190648 | nM | Homo sapiens |