# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4209136 | 22 | F | = | 50.3 | % | ALA4184710 | % | Rattus norvegicus | |||
2. | ALA4209136 | 22 | Vdss | = | 5.9 | L/Kg | ALA4184709 | L.kg-1 | Rattus norvegicus | |||
3. | ALA4209136 | 22 | CL | = | 72 | ml/min.kg | ALA4184708 | mL.min-1.kg-1 | Rattus norvegicus | |||
4. | ALA4209136 | 22 | t1/2 | = | 1.9 | hr | ALA4184706 | hr | Rattus norvegicus | |||
5. | ALA4209136 | 22 | t1/2 | = | 3.3 | hr | ALA4184705 | hr | Rattus norvegicus | |||
6. | ALA4209136 | 22 | Cmax | = | 356 | ng/ml | ALA4184704 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
7. | ALA4209136 | 22 | t1/2 | = | 122 | min | ALA4184703 | hr | ||||
8. | ALA4209136 | 22 | t1/2 | = | 52 | min | ALA4184702 | hr | ||||
9. | ALA4209136 | 22 | EC50 | = | 6 | nM | ALA4184699 | 8.22 | nM | Rattus norvegicus | ||
10. | ALA4209136 | 22 | EC50 | = | 30 | nM | ALA4184698 | 7.52 | nM | Homo sapiens |