| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4209316 | BMS-932481 | EC50 | = | 7 | nM | ALA4431691 | 8.15 | nM | Homo sapiens | ||
| 2. | ALA4209316 | BMS-932481 | Drug metabolism | 0 | ALA4701736 | Metabolite_Detected | ||||||
| 3. | ALA4209316 | BMS-932481 | Kinact | = | 0.47 | /min | ALA4701735 | /min | Homo sapiens | |||
| 4. | ALA4209316 | BMS-932481 | Ki | = | 82.5 | uM | ALA4701734 | 4.08 | nM | Homo sapiens | ||
| 5. | ALA4209316 | BMS-932481 | Drug metabolism | 0 | ALA4701733 | Metabolite_Detected | ||||||
| 6. | ALA4209316 | BMS-932481 | Drug metabolism | 0 | ALA4701732 | Not Active | ||||||
| 7. | ALA4209316 | BMS-932481 | Drug metabolism | 0 | ALA4701731 | Metabolite_Detected | ||||||
| 8. | ALA4209316 | BMS-932481 | Drug metabolism | 0 | ALA4701730 | Metabolite_Detected | ||||||
| 9. | ALA4209316 | BMS-932481 | Stabilty | = | 89 | % | ALA4701729 | % | ||||
| 10. | ALA4209316 | BMS-932481 | Stabilty | = | 94 | % | ALA4701728 | % | ||||
| 11. | ALA4209316 | BMS-932481 | IC50 | = | 4 | nM | ALA4701727 | 8.40 | nM | Homo sapiens | ||
| 12. | ALA4209316 | BMS-932481 | Activity | 0 | ALA4700856 | Non-Toxic | ||||||
| 13. | ALA4209316 | BMS-932481 | Activity | 0 | ALA4700855 | Non-Toxic | ||||||
| 14. | ALA4209316 | BMS-932481 | Activity | 0 | ALA4700854 | Toxic | ||||||
| 15. | ALA4209316 | BMS-932481 | NOAEL | = | 150 | mg kg-1 | ALA4700853 | mg kg-1 | ||||
| 16. | ALA4209316 | BMS-932481 | AUC | = | 180 | uM.hr | ALA4700852 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 17. | ALA4209316 | BMS-932481 | Cmax | = | 14 | uM | ALA4700851 | nM | ||||
| 18. | ALA4209316 | BMS-932481 | Activity | 0 | ALA4700850 | Non-Toxic | ||||||
| 19. | ALA4209316 | BMS-932481 | Activity | 0 | ALA4700849 | Non-Toxic | ||||||
| 20. | ALA4209316 | BMS-932481 | Activity | 0 | ALA4700848 | Non-Toxic |
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