| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4209341 | 27e | Activity | 0 | ALA4184894 | Active | Mus musculus | |||||
| 2. | ALA4209341 | 27e | Activity | 0 | ALA4184893 | Active | Mus musculus | |||||
| 3. | ALA4209341 | 27e | permeability | 0 | ALA4184891 | Permeable | ||||||
| 4. | ALA4209341 | 27e | AUC | = | 19187 | nM.hr | ALA4184886 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 5. | ALA4209341 | 27e | AUC | = | 6183 | nM.hr | ALA4184885 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 6. | ALA4209341 | 27e | F | = | 31 | % | ALA4184884 | % | Mus musculus | |||
| 7. | ALA4209341 | 27e | Tmax | = | 0.5 | hr | ALA4184883 | hr | Mus musculus | |||
| 8. | ALA4209341 | 27e | Cmax | = | 12691 | nM | ALA4184882 | nM | Mus musculus | |||
| 9. | ALA4209341 | 27e | Vdss | = | 0.5 | L/Kg | ALA4184881 | L.kg-1 | Mus musculus | |||
| 10. | ALA4209341 | 27e | t1/2 | = | 1.5 | hr | ALA4184874 | hr | Mus musculus | |||
| 11. | ALA4209341 | 27e | CL | = | 6.8 | ml/min.kg | ALA4184875 | mL.min-1.kg-1 | Mus musculus | |||
| 12. | ALA4209341 | 27e | T/C | = | 0.48 | ALA4184879 | Homo sapiens | |||||
| 13. | ALA4209341 | 27e | INH | = | 17.1 | uM | ALA4184872 | uM | Homo sapiens | |||
| 14. | ALA4209341 | 27e | solubility | < | 0.004 | mM | ALA4184873 | nM | ||||
| 15. | ALA4209341 | 27e | IC50 | = | 8 | nM | ALA4184877 | 8.10 | nM | Homo sapiens | ||
| 16. | ALA4209341 | 27e | IC50 | = | 1 | nM | ALA4184876 | 9.00 | nM | Homo sapiens | ||
| 17. | ALA4209341 | 27e | CLH | = | 148 | microL/min/mg | ALA4184895 | mL.min-1.g-1 |
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