# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4209981 | 10h | Activity | 0 | ALA4198067 | Not Active | Homo sapiens | |||||
2. | ALA4209981 | 10h | Activity | 0 | ALA4198066 | Not Active | Homo sapiens | |||||
3. | ALA4209981 | 10h | Activity | 0 | ALA4198065 | Not Active | Homo sapiens | |||||
4. | ALA4209981 | 10h | Activity | 0 | ALA4198064 | Dose-dependent effect | Homo sapiens | |||||
5. | ALA4209981 | 10h | CLH | = | 9.6 | ml/min.kg | ALA4198063 | mL.min-1.kg-1 | ||||
6. | ALA4209981 | 10h | t1/2 | = | 2.16 | hr | ALA4198062 | hr | ||||
7. | ALA4209981 | 10h | CLH | = | 39 | ml/min.kg | ALA4198061 | mL.min-1.kg-1 | ||||
8. | ALA4209981 | 10h | t1/2 | = | 1.2 | hr | ALA4198060 | hr | ||||
9. | ALA4209981 | 10h | CLH | = | 48.7 | ml/min.kg | ALA4198059 | mL.min-1.kg-1 | ||||
10. | ALA4209981 | 10h | t1/2 | = | 1.17 | hr | ALA4198058 | hr | ||||
11. | ALA4209981 | 10h | Ratio IC50 | = | 0.32 | ALA4198057 | ||||||
12. | ALA4209981 | 10h | Ratio IC50 | = | 0.13 | ALA4198056 | ||||||
13. | ALA4209981 | 10h | IC50 | = | 0.06 | uM | ALA4198055 | 7.22 | nM | Homo sapiens | ||
14. | ALA4209981 | 10h | IC50 | = | 0.19 | uM | ALA4198054 | 6.72 | nM | Homo sapiens | ||
15. | ALA4209981 | 10h | IC50 | = | 0.18 | uM | ALA4198053 | 6.75 | nM | |||
16. | ALA4209981 | 10h | IC50 | = | 1.39 | uM | ALA4198052 | 5.86 | nM | Homo sapiens | ||
17. | ALA4209981 | 10h | Ratio IC50 | 0 | ALA4198051 | Not Determined | ||||||
18. | ALA4209981 | 10h | IC50 | = | 2.2 | uM | ALA4198050 | 5.66 | nM | |||
19. | ALA4209981 | 10h | IC50 | 0 | ALA4198049 | Not Determined | Homo sapiens | |||||
20. | ALA4209981 | 10h | IC50 | = | 3.7 | uM | ALA4198048 | 5.43 | nM | Homo sapiens |