| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4212095 | 5 | IC50 | = | 61 | nM | ALA4199684 | 7.21 | nM | Homo sapiens | ||
| 2. | ALA4212095 | 5 | IC50 | = | 16 | nM | ALA4199685 | 7.80 | nM | Homo sapiens | ||
| 3. | ALA4212095 | 5 | IC50 | > | 90000 | nM | ALA4199686 | nM | Homo sapiens | |||
| 4. | ALA4212095 | 5 | INH | 0 | ALA4199687 | Active | % | Homo sapiens | ||||
| 5. | ALA4212095 | 5 | pKa | = | 6.5 | ALA4199688 | ||||||
| 6. | ALA4212095 | 5 | Cmax | = | 25 | uM | ALA4199689 | nM | Mus musculus | |||
| 7. | ALA4212095 | 5 | AUC | = | 19 | uM.hr | ALA4199690 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 8. | ALA4212095 | 5 | CL | = | 2.5 | ml/min.kg | ALA4199691 | mL.min-1.kg-1 | Mus musculus | |||
| 9. | ALA4212095 | 5 | t1/2 | = | 4.9 | hr | ALA4199692 | hr | Mus musculus | |||
| 10. | ALA4212095 | 5 | Cmax | = | 2 | uM | ALA4199693 | nM | Mus musculus | |||
| 11. | ALA4212095 | 5 | AUC | = | 16 | uM.hr | ALA4199694 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Mus musculus | ||
| 12. | ALA4212095 | 5 | t1/2 | = | 2.9 | hr | ALA4199695 | hr | Mus musculus | |||
| 13. | ALA4212095 | 5 | F | = | 82 | % | ALA4199696 | % | Mus musculus |
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