# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4212186 | 44b; CM-407 | IC50 | = | 11 | nM | ALA4268472 | 7.96 | nM | Homo sapiens | ||
2. | ALA4212186 | 44b; CM-407 | Activity | = | 68 | % | ALA4198947 | % | Mus musculus | |||
3. | ALA4212186 | 44b; CM-407 | Activity | = | 48 | % | ALA4198946 | % | Mus musculus | |||
4. | ALA4212186 | 44b; CM-407 | IC50 | > | 10 | uM | ALA4198945 | nM | Homo sapiens | |||
5. | ALA4212186 | 44b; CM-407 | IC50 | > | 10 | uM | ALA4198944 | nM | Homo sapiens | |||
6. | ALA4212186 | 44b; CM-407 | IC50 | > | 10 | uM | ALA4198943 | nM | Homo sapiens | |||
7. | ALA4212186 | 44b; CM-407 | IC50 | > | 10 | uM | ALA4198942 | nM | Homo sapiens | |||
8. | ALA4212186 | 44b; CM-407 | IC50 | = | 3.2 | uM | ALA4198941 | 5.50 | nM | Homo sapiens | ||
9. | ALA4212186 | 44b; CM-407 | IC50 | = | 1.4 | nM | ALA4198940 | 8.85 | nM | Homo sapiens | ||
10. | ALA4212186 | 44b; CM-407 | IC50 | > | 10 | uM | ALA4198939 | nM | Homo sapiens | |||
11. | ALA4212186 | 44b; CM-407 | t1/2 | = | 5.2 | min | ALA4198938 | hr | ||||
12. | ALA4212186 | 44b; CM-407 | t1/2 | = | 32.7 | min | ALA4198937 | hr | ||||
13. | ALA4212186 | 44b; CM-407 | INH | = | 23.4 | % | ALA4198936 | % | Homo sapiens | |||
14. | ALA4212186 | 44b; CM-407 | INH | < | 50 | % | ALA4198935 | % | Homo sapiens | |||
15. | ALA4212186 | 44b; CM-407 | INH | < | 50 | % | ALA4198934 | % | Homo sapiens | |||
16. | ALA4212186 | 44b; CM-407 | INH | < | 50 | % | ALA4198933 | % | Homo sapiens | |||
17. | ALA4212186 | 44b; CM-407 | INH | < | 50 | % | ALA4198932 | % | Homo sapiens | |||
18. | ALA4212186 | 44b; CM-407 | LC50 | = | 46300 | nM | ALA4198931 | nM | Mus musculus | |||
19. | ALA4212186 | 44b; CM-407 | INH | = | 30 | % | ALA4198930 | % | Mus musculus | |||
20. | ALA4212186 | 44b; CM-407 | INH | = | 55 | % | ALA4198929 | % | Mus musculus |