# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4214738 | 15r; VU6008541 | pEC50 | = | 6.51 | ALA4180102 | 6.51 | nM | Rattus norvegicus | |||
2. | ALA4214738 | 15r; VU6008541 | K(p,uu,brain) | = | 0.3 | ALA4180112 | ||||||
3. | ALA4214738 | 15r; VU6008541 | Kp | = | 0.1 | ALA4180111 | ||||||
4. | ALA4214738 | 15r; VU6008541 | Fu | = | 0.006 | ALA4180110 | ||||||
5. | ALA4214738 | 15r; VU6008541 | Fu | = | 0.002 | ALA4180109 | ||||||
6. | ALA4214738 | 15r; VU6008541 | Fu | = | 0.002 | ALA4180108 | ||||||
7. | ALA4214738 | 15r; VU6008541 | CLH | = | 18.6 | ml/min.kg | ALA4180107 | mL.min-1.kg-1 | ||||
8. | ALA4214738 | 15r; VU6008541 | CLH | = | 160 | ml/min.kg | ALA4180106 | mL.min-1.kg-1 | ||||
9. | ALA4214738 | 15r; VU6008541 | CLH | = | 56.6 | ml/min.kg | ALA4180105 | mL.min-1.kg-1 | ||||
10. | ALA4214738 | 15r; VU6008541 | CLH | = | 295 | ml/min.kg | ALA4180104 | mL.min-1.kg-1 | ||||
11. | ALA4214738 | 15r; VU6008541 | %max | = | 57 | % | ALA4180103 | % | Rattus norvegicus | |||
12. | ALA4214738 | 15r; VU6008541 | EC50 | = | 307 | nM | ALA4180102 | 6.51 | nM | Rattus norvegicus |