# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4216791 | 14 | Drug recovery | = | 92 | % | ALA4179238 | % | ||||
2. | ALA4216791 | 14 | Drug recovery | = | 100 | % | ALA4179237 | % | ||||
3. | ALA4216791 | 14 | Drug recovery | = | 96 | % | ALA4179236 | % | ||||
4. | ALA4216791 | 14 | Drug recovery | = | 90 | % | ALA4179235 | % | ||||
5. | ALA4216791 | 14 | Drug recovery | = | 91 | % | ALA4179234 | % | ||||
6. | ALA4216791 | 14 | Drug recovery | = | 100 | % | ALA4179233 | % | ||||
7. | ALA4216791 | 14 | t1/2 | > | 30 | min | ALA4179232 | hr | ||||
8. | ALA4216791 | 14 | t1/2 | > | 30 | min | ALA4179231 | hr | ||||
9. | ALA4216791 | 14 | t1/2 | > | 30 | min | ALA4179228 | hr | ||||
10. | ALA4216791 | 14 | Drug metabolism | < | 0.04 | nmol/min/mg | ALA4179230 | nmol/min/mg | ||||
11. | ALA4216791 | 14 | Drug metabolism | < | 0.04 | nmol/min/mg | ALA4179229 | nmol/min/mg | ||||
12. | ALA4216791 | 14 | Drug metabolism | < | 0.04 | nmol/min/mg | ALA4179227 | nmol/min/mg | ||||
13. | ALA4216791 | 14 | Ki | = | 2.7 | nM | ALA4179226 | 8.57 | nM | Bos taurus |