# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4225470 | 10 | INH | 0 | ALA4219880 | Active | % | Homo sapiens | ||||
2. | ALA4225470 | 10 | t1/2 | = | 7.073 | s | ALA4219897 | hr | Homo sapiens | |||
3. | ALA4225470 | 10 | Kd | = | 16 | nM | ALA4219896 | 7.80 | nM | Homo sapiens | ||
4. | ALA4225470 | 10 | K | = | 0.098 | /s | ALA4219895 | /s | Homo sapiens | |||
5. | ALA4225470 | 10 | K | = | 5.99 | 10'5/M/s | ALA4219894 | 10'5/M/s | Homo sapiens | |||
6. | ALA4225470 | 10 | CLH | = | 2.9 | ml/min/g | ALA4219893 | mL.min-1.g-1 | ||||
7. | ALA4225470 | 10 | t1/2 | > | 180 | min | ALA4219892 | hr | ||||
8. | ALA4225470 | 10 | t1/2 | = | 11.94 | s | ALA4219891 | hr | Homo sapiens | |||
9. | ALA4225470 | 10 | Kd | = | 24 | nM | ALA4219890 | 7.62 | nM | Homo sapiens | ||
10. | ALA4225470 | 10 | K | = | 0.058 | /s | ALA4219889 | /s | Homo sapiens | |||
11. | ALA4225470 | 10 | K | = | 2.4 | 10'6/M/s | ALA4219888 | 10'6/M/s | Homo sapiens | |||
12. | ALA4225470 | 10 | logD | = | 1.63 | ALA4219887 | ||||||
13. | ALA4225470 | 10 | permeability | = | 27.1 | nm/s | ALA4219886 | nm/s | ||||
14. | ALA4225470 | 10 | Activity | 0 | ALA4219885 | Toxic | Homo sapiens | |||||
15. | ALA4225470 | 10 | Activity | 0 | ALA4219884 | Toxic | Homo sapiens | |||||
16. | ALA4225470 | 10 | Activity | = | 175 | % | ALA4219883 | % | Homo sapiens | |||
17. | ALA4225470 | 10 | Kd | = | 44 | nM | ALA4219882 | 7.36 | nM | Homo sapiens | ||
18. | ALA4225470 | 10 | Kd | = | 90 | nM | ALA4219881 | 7.05 | nM | Homo sapiens |