# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | VH 298 | 15; VH298 | Activity | 0 | ALA5225297 | Active | Homo sapiens | |||||
2. | VH 298 | 15; VH298 | Activity | 0 | ALA5225296 | Not Active | Homo sapiens | |||||
3. | VH 298 | 15; VH298 | Kd | = | 90 | nM | ALA4396995 | 7.05 | nM | Homo sapiens | ||
4. | VH 298 | 15; VH298 | Kd | = | 58 | nM | ALA4730314 | 7.24 | nM | Homo sapiens | ||
5. | VH 298 | 15; VH298 | t1/2 | = | 5.874 | s | ALA4219897 | hr | Homo sapiens | |||
6. | VH 298 | 15; VH298 | Kd | = | 52 | nM | ALA4219896 | 7.28 | nM | Homo sapiens | ||
7. | VH 298 | 15; VH298 | K | = | 0.118 | /s | ALA4219895 | /s | Homo sapiens | |||
8. | VH 298 | 15; VH298 | K | = | 7.8 | 10'5/M/s | ALA4219894 | 10'5/M/s | Homo sapiens | |||
9. | VH 298 | 15; VH298 | CLH | = | 3.1 | ml/min/g | ALA4219893 | mL.min-1.g-1 | ||||
10. | VH 298 | 15; VH298 | t1/2 | > | 180 | min | ALA4219892 | hr | ||||
11. | VH 298 | 15; VH298 | t1/2 | = | 10.66 | s | ALA4219891 | hr | Homo sapiens | |||
12. | VH 298 | 15; VH298 | Kd | = | 99 | nM | ALA4219890 | 7.00 | nM | Homo sapiens | ||
13. | VH 298 | 15; VH298 | K | = | 0.065 | /s | ALA4219889 | /s | Homo sapiens | |||
14. | VH 298 | 15; VH298 | K | = | 6.6 | 10'5/M/s | ALA4219888 | 10'5/M/s | Homo sapiens | |||
15. | VH 298 | 15; VH298 | logD | = | 1.4 | ALA4219887 | ||||||
16. | VH 298 | 15; VH298 | permeability | = | 19.4 | nm/s | ALA4219886 | nm/s | ||||
17. | VH 298 | 15; VH298 | Activity | 0 | ALA4219885 | Non-Toxic | Homo sapiens | |||||
18. | VH 298 | 15; VH298 | Activity | 0 | ALA4219884 | Non-Toxic | Homo sapiens | |||||
19. | VH 298 | 15; VH298 | Activity | = | 190 | % | ALA4219883 | % | Homo sapiens | |||
20. | VH 298 | 15; VH298 | Kd | = | 90 | nM | ALA4219882 | 7.05 | nM | Homo sapiens |