| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4227228 | MK-3901 | t1/2 | = | 1 | hr | ALA4222594 | hr | Rattus norvegicus | |||
| 2. | ALA4227228 | MK-3901 | CL | = | 133 | ml/min.kg | ALA4222593 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 3. | ALA4227228 | MK-3901 | PPB | = | 98.4 | % | ALA4222592 | % | ||||
| 4. | ALA4227228 | MK-3901 | F | = | 47 | % | ALA4222591 | % | Macaca mulatta | |||
| 5. | ALA4227228 | MK-3901 | F | = | 68 | % | ALA4222590 | % | Canis lupus familiaris | |||
| 6. | ALA4227228 | MK-3901 | F | = | 60 | % | ALA4222589 | % | Rattus norvegicus | |||
| 7. | ALA4227228 | MK-3901 | IC50 | = | 1 | uM | ALA4222588 | 6.00 | nM | Homo sapiens | ||
| 8. | ALA4227228 | MK-3901 | Activity | = | 47 | % | ALA4222587 | % | Homo sapiens | |||
| 9. | ALA4227228 | MK-3901 | IC50 | = | 5.7 | uM | ALA4222586 | 5.24 | nM | Homo sapiens | ||
| 10. | ALA4227228 | MK-3901 | EC90 | = | 3 | uM | ALA4222585 | uM | Rattus norvegicus | |||
| 11. | ALA4227228 | MK-3901 | IC50 | = | 24 | nM | ALA4222584 | 7.62 | nM | Homo sapiens | ||
| 12. | ALA4227228 | MK-3901 | INH | = | 21 | nM | ALA4222583 | nM | Homo sapiens |
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