# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4227834 | 8; MZP-61 | Peff | = | 0.3 | 10^-6 cm/s | ALA4730316 | 10^-6 cm/s | ||||
2. | ALA4227834 | 8; MZP-61 | logD | = | -0.7 | ALA4730315 | ||||||
3. | ALA4227834 | 8; MZP-61 | Kd | = | 781 | nM | ALA4219529 | 6.11 | nM | Homo sapiens | ||
4. | ALA4227834 | 8; MZP-61 | Kd | = | 116 | nM | ALA4219528 | 6.94 | nM | Homo sapiens | ||
5. | ALA4227834 | 8; MZP-61 | Kd | = | 3 | nM | ALA4219527 | 8.52 | nM | Homo sapiens | ||
6. | ALA4227834 | 8; MZP-61 | Activity | = | 14 | % | ALA4219526 | % | Homo sapiens | |||
7. | ALA4227834 | 8; MZP-61 | Activity | = | -156 | % | ALA4219525 | % | Homo sapiens | |||
8. | ALA4227834 | 8; MZP-61 | Activity | = | 11 | % | ALA4219524 | % | Homo sapiens | |||
9. | ALA4227834 | 8; MZP-61 | Activity | = | 11 | % | ALA4219517 | % | Homo sapiens | |||
10. | ALA4227834 | 8; MZP-61 | Emax | = | 96.6 | % | ALA4219518 | % | Homo sapiens | |||
11. | ALA4227834 | 8; MZP-61 | Emax | = | 88.1 | % | ALA4219523 | % | Homo sapiens | |||
12. | ALA4227834 | 8; MZP-61 | pEC50 | = | 6.17 | ALA4219518 | 6.17 | nM | Homo sapiens | |||
13. | ALA4227834 | 8; MZP-61 | pEC50 | = | 6.24 | ALA4219523 | 6.24 | nM | Homo sapiens | |||
14. | ALA4227834 | 8; MZP-61 | Emax | = | 37 | % | ALA4219522 | % | Homo sapiens | |||
15. | ALA4227834 | 8; MZP-61 | Emax | = | 74 | % | ALA4219521 | % | Homo sapiens | |||
16. | ALA4227834 | 8; MZP-61 | Emax | = | 78 | % | ALA4219520 | % | ||||
17. | ALA4227834 | 8; MZP-61 | pDC50 | = | 6.8 | ALA4219515 | Homo sapiens | |||||
18. | ALA4227834 | 8; MZP-61 | pDC50 | = | 6.7 | ALA4219514 | ||||||
19. | ALA4227834 | 8; MZP-61 | pDC50 | = | 6.9 | ALA4219513 | ||||||
20. | ALA4227834 | 8; MZP-61 | Emax | = | 94 | % | ALA4219519 | % |