| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4228478 | 4 | IC50 | = | 5 | nM | ALA4222142 | 8.30 | nM | Homo sapiens | ||
| 2. | ALA4228478 | 4 | IC50 | = | 124 | nM | ALA4222141 | 6.91 | nM | Homo sapiens | ||
| 3. | ALA4228478 | 4 | Ratio IC50 | > | 1000 | ALA4222143 | ||||||
| 4. | ALA4228478 | 4 | Ratio IC50 | > | 1000 | ALA4222144 | ||||||
| 5. | ALA4228478 | 4 | Ratio IC50 | > | 1000 | ALA4222145 | ||||||
| 6. | ALA4228478 | 4 | Ratio IC50 | > | 1000 | ALA4222146 | ||||||
| 7. | ALA4228478 | 4 | Ratio IC50 | > | 1000 | ALA4222147 | ||||||
| 8. | ALA4228478 | 4 | Ratio IC50 | > | 1000 | ALA4222148 | ||||||
| 9. | ALA4228478 | 4 | Ratio IC50 | > | 1000 | ALA4222149 | ||||||
| 10. | ALA4228478 | 4 | Ratio IC50 | > | 1000 | ALA4222150 | ||||||
| 11. | ALA4228478 | 4 | Ratio IC50 | > | 1000 | ALA4222151 | ||||||
| 12. | ALA4228478 | 4 | Ratio IC50 | = | 1189 | ALA4222152 | ||||||
| 13. | ALA4228478 | 4 | CL | = | 19 | ml/min.kg | ALA4222153 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 14. | ALA4228478 | 4 | t1/2 | = | 4.7 | hr | ALA4222154 | hr | Rattus norvegicus | |||
| 15. | ALA4228478 | 4 | Vdss | = | 3.6 | L/Kg | ALA4222155 | L.kg-1 | Rattus norvegicus | |||
| 16. | ALA4228478 | 4 | F | = | 30 | % | ALA4222156 | % | Rattus norvegicus | |||
| 17. | ALA4228478 | 4 | PPB | = | 98 | % | ALA4222157 | % | ||||
| 18. | ALA4228478 | 4 | Activity | 0 | ALA4222158 | Dose-dependent effect | Rattus norvegicus | |||||
| 19. | ALA4228478 | 4 | Activity | = | 15 | % | ALA4222159 | % | Rattus norvegicus | |||
| 20. | ALA4228478 | 4 | Cp | = | 0.05 | uM | ALA4222160 | uM | Rattus norvegicus |
The page will load shortly, Thanks for your patience!