| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4228859 | 9 | INH | 0 | ALA4221510 | Dose-dependent effect | % | Mus musculus | ||||
| 2. | ALA4228859 | 9 | IC50 | = | 3.8 | uM | ALA4221509 | 5.42 | nM | Homo sapiens | ||
| 3. | ALA4228859 | 9 | INH | < | 20 | % | ALA4221508 | % | Homo sapiens | |||
| 4. | ALA4228859 | 9 | INH | < | 20 | % | ALA4221507 | % | Homo sapiens | |||
| 5. | ALA4228859 | 9 | INH | < | 20 | % | ALA4221506 | % | Homo sapiens | |||
| 6. | ALA4228859 | 9 | INH | < | 20 | % | ALA4221505 | % | Homo sapiens | |||
| 7. | ALA4228859 | 9 | INH | < | 20 | % | ALA4221488 | % | Homo sapiens | |||
| 8. | ALA4228859 | 9 | Fu | = | 32 | % | ALA4221504 | |||||
| 9. | ALA4228859 | 9 | BPR | = | 0.4 | ALA4221503 | ||||||
| 10. | ALA4228859 | 9 | F | = | 105 | % | ALA4221502 | % | Rattus norvegicus | |||
| 11. | ALA4228859 | 9 | Tmax | = | 1 | hr | ALA4221501 | hr | Rattus norvegicus | |||
| 12. | ALA4228859 | 9 | Cmax | = | 2452 | nM | ALA4221500 | nM | Rattus norvegicus | |||
| 13. | ALA4228859 | 9 | BPR | = | 0.2 | ALA4221499 | ||||||
| 14. | ALA4228859 | 9 | t1/2 | = | 3.1 | hr | ALA4221498 | hr | Rattus norvegicus | |||
| 15. | ALA4228859 | 9 | Vdss | = | 1.8 | L/Kg | ALA4221497 | L.kg-1 | Rattus norvegicus | |||
| 16. | ALA4228859 | 9 | CL | = | 32 | ml/min.kg | ALA4221496 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 17. | ALA4228859 | 9 | Fu | = | 14 | % | ALA4221495 | |||||
| 18. | ALA4228859 | 9 | CLH | = | 182 | microL/min/mg | ALA4221494 | mL.min-1.g-1 | ||||
| 19. | ALA4228859 | 9 | Ratio | = | 6.2 | ALA4221493 | ||||||
| 20. | ALA4228859 | 9 | CLH | = | 121 | microL/min/mg | ALA4221492 | mL.min-1.g-1 |
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