# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4237449 | 10 | Ratio | = | 0.5 | ALA4344590 | Homo sapiens | |||||
2. | ALA4237449 | 10 | FC | = | 1.4 | ALA4344589 | Homo sapiens | |||||
3. | ALA4237449 | 10 | -TdeltaS | = | 5.71 | kcal/mol | ALA4344581 | kcal/mol | Homo sapiens | |||
4. | ALA4237449 | 10 | deltaH | = | -12.2 | kcal/mol | ALA4344580 | kcal/mol | Homo sapiens | |||
5. | ALA4237449 | 10 | deltaG | = | -6.5 | kcal/mol | ALA4344579 | kcal/mol | Homo sapiens | |||
6. | ALA4237449 | 10 | Kd | = | 16.9 | uM | ALA4344578 | 4.77 | nM | Homo sapiens | ||
7. | ALA4237449 | 10 | EC50 | = | 0.3 | uM | ALA4344577 | 6.52 | nM | Homo sapiens | ||
8. | ALA4237449 | 10 | INH | = | 10 | % | ALA4344576 | % | Homo sapiens | |||
9. | ALA4237449 | 10 | Ratio EC50 | > | 20 | ALA4344575 | ||||||
10. | ALA4237449 | 10 | Ratio EC50 | > | 20 | ALA4344574 | ||||||
11. | ALA4237449 | 10 | EC50 | > | 100 | uM | ALA4344573 | nM | Homo sapiens | |||
12. | ALA4237449 | 10 | EC50 | > | 100 | uM | ALA4344572 | nM | Homo sapiens | |||
13. | ALA4237449 | 10 | EC50 | = | 4.43 | uM | ALA4344571 | 5.35 | nM | Homo sapiens | ||
14. | ALA4237449 | 10 | Activity | 0 | ALA4344570 | Non-Toxic | ||||||
15. | ALA4237449 | 10 | Activity | = | 4.68 | % | ALA4344568 | % | ||||
16. | ALA4237449 | 10 | Activity | = | 0.062 | ug | ALA4344567 | ug | Rattus norvegicus | |||
17. | ALA4237449 | 10 | Activity | 0 | ALA4344565 | Non-Toxic | Mus musculus | |||||
18. | ALA4237449 | 10 | INH | 0 | ALA4344564 | Not Active | % | Homo sapiens | ||||
19. | ALA4237449 | 10 | INH | 0 | ALA4344563 | Not Active | % | Homo sapiens | ||||
20. | ALA4237449 | 10 | INH | 0 | ALA4344562 | Not Active | % | Homo sapiens |