| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4242598 | 16 | IC50 | = | 0.7 | nM | ALA4236252 | 9.15 | nM | Homo sapiens | ||
| 2. | ALA4242598 | 16 | permeability | = | 6.7 | 10'-6 cm/s | ALA4236253 | 10'-6 cm/s | ||||
| 3. | ALA4242598 | 16 | Ratio | = | 6.1 | ALA4236254 | ||||||
| 4. | ALA4242598 | 16 | CLH | = | 74 | uL/min | ALA4236255 | uL/min | ||||
| 5. | ALA4242598 | 16 | CLH | = | 62 | uL/min | ALA4236256 | uL/min | ||||
| 6. | ALA4242598 | 16 | CLH | = | 203 | uL/min | ALA4236257 | uL/min | ||||
| 7. | ALA4242598 | 16 | IC50 | = | 9.7 | nM | ALA4236258 | 8.01 | nM | Homo sapiens | ||
| 8. | ALA4242598 | 16 | IC50 | = | 82 | nM | ALA4236259 | 7.09 | nM | Homo sapiens | ||
| 9. | ALA4242598 | 16 | Fu | = | 0.46 | % | ALA4236260 | |||||
| 10. | ALA4242598 | 16 | Fu | = | 0.2 | % | ALA4236261 | |||||
| 11. | ALA4242598 | 16 | Fu | = | 0.31 | % | ALA4236262 | |||||
| 12. | ALA4242598 | 16 | Ki | = | 2.2 | uM | ALA4236263 | 5.66 | nM | Homo sapiens | ||
| 13. | ALA4242598 | 16 | IC50 | = | 0.1 | uM | ALA4236264 | 7.00 | nM | Homo sapiens | ||
| 14. | ALA4242598 | 16 | CL | = | 1.24 | L/hr/kg | ALA4236269 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 15. | ALA4242598 | 16 | Vdss | = | 0.86 | L/Kg | ALA4236270 | L.kg-1 | Rattus norvegicus | |||
| 16. | ALA4242598 | 16 | t1/2 | = | 0.72 | hr | ALA4236271 | hr | Rattus norvegicus | |||
| 17. | ALA4242598 | 16 | F | = | 47 | % | ALA4236272 | % | Rattus norvegicus | |||
| 18. | ALA4242598 | 16 | INH | = | 98 | % | ALA4236273 | % | Homo sapiens | |||
| 19. | ALA4242598 | 16 | INH | = | 96 | % | ALA4236274 | % | Homo sapiens | |||
| 20. | ALA4242598 | 16 | INH | = | 95 | % | ALA4236275 | % | Homo sapiens |
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