# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4242635 | 28b; 8 Isomer 2B | Activity | 0 | ALA4236990 | Dose-dependent effect | ||||||
2. | ALA4242635 | 28b; 8 Isomer 2B | Selectivity ratio | = | 0.2 | ALA4236911 | ||||||
3. | ALA4242635 | 28b; 8 Isomer 2B | Selectivity ratio | = | 0.3 | ALA4236910 | ||||||
4. | ALA4242635 | 28b; 8 Isomer 2B | Selectivity ratio | = | 1.6 | ALA4236909 | ||||||
5. | ALA4242635 | 28b; 8 Isomer 2B | Selectivity ratio | = | 1.6 | ALA4236908 | ||||||
6. | ALA4242635 | 28b; 8 Isomer 2B | logD | = | 3.34 | ALA4236907 | ||||||
7. | ALA4242635 | 28b; 8 Isomer 2B | pIC50 | = | 5.7 | ALA4236906 | 5.70 | nM | Homo sapiens | |||
8. | ALA4242635 | 28b; 8 Isomer 2B | pIC50 | = | 5.3 | ALA4236905 | 5.30 | nM | Homo sapiens | |||
9. | ALA4242635 | 28b; 8 Isomer 2B | pKi | = | 10.1 | ALA4236904 | 10.10 | nM | Homo sapiens | |||
10. | ALA4242635 | 28b; 8 Isomer 2B | pIC50 | = | 8.2 | ALA4236903 | 8.20 | nM | Homo sapiens | |||
11. | ALA4242635 | 28b; 8 Isomer 2B | pIC50 | = | 8.4 | ALA4236899 | 8.40 | nM | Homo sapiens | |||
12. | ALA4242635 | 28b; 8 Isomer 2B | pIC50 | = | 6.8 | ALA4236900 | 6.80 | nM | Homo sapiens | |||
13. | ALA4242635 | 28b; 8 Isomer 2B | pIC50 | = | 6.8 | ALA4236902 | 6.80 | nM | Homo sapiens | |||
14. | ALA4242635 | 28b; 8 Isomer 2B | pIC50 | = | 8.1 | ALA4236901 | 8.10 | nM | Homo sapiens |