# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4246000 | M3 | Kd | = | 197.8 | nM | ALA4234630 | 6.70 | nM | Homo sapiens | ||
2. | ALA4246000 | M3 | K | = | 45.3 | 10'-3/s | ALA4234631 | 10'-3/s | Homo sapiens | |||
3. | ALA4246000 | M3 | K | = | 2.29 | 10'5/M/s | ALA4234632 | 10'5/M/s | Homo sapiens | |||
4. | ALA4246000 | M3 | t1/2 | = | 15.3 | s | ALA4234633 | hr | Homo sapiens | |||
5. | ALA4246000 | M3 | Papp | = | 0.3 | 10'-6 cm/s | ALA4234634 | 10'-6 cm/s | ||||
6. | ALA4246000 | M3 | logD | = | 0.08 | ALA4234635 | ||||||
7. | ALA4246000 | M3 | Activity | 0 | ALA4234636 | Not Determined | Homo sapiens | |||||
8. | ALA4246000 | M3 | Activity | 0 | ALA4234637 | Not Determined | Homo sapiens | |||||
9. | ALA4246000 | M3 | Activity | 0 | ALA4234638 | Not Determined | Homo sapiens | |||||
10. | ALA4246000 | M3 | Activity | = | 147 | % | ALA4234639 | % | Homo sapiens | |||
11. | ALA4246000 | M3 | Activity | = | 193 | % | ALA4234640 | % | Homo sapiens | |||
12. | ALA4246000 | M3 | EC50 | > | 40000 | nM | ALA4234621 | nM | Homo sapiens | |||
13. | ALA4246000 | M3 | EC50 | > | 40000 | nM | ALA4234641 | nM | Homo sapiens | |||
14. | ALA4246000 | M3 | EC50 | > | 40000 | nM | ALA4234642 | nM | Homo sapiens | |||
15. | ALA4246000 | M3 | EC50 | = | 332 | nM | ALA4234643 | 6.48 | nM | Homo sapiens | ||
16. | ALA4246000 | M3 | EC50 | = | 59 | nM | ALA4234644 | 7.23 | nM | Homo sapiens | ||
17. | ALA4246000 | M3 | t1/2 | > | 21 | hr | ALA4234645 | hr | ||||
18. | ALA4246000 | M3 | Retention_time | = | 8.37 | min | ALA4234646 | min | Homo sapiens | |||
19. | ALA4246000 | M3 | Drug metabolism | 0 | ALA4234648 | Metabolite_Detected |