# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4248974 | 19 | Activity | = | 154 | mm3 | ALA4235129 | mm3 | Homo sapiens | |||
2. | ALA4248974 | 19 | solubility | = | 28.2 | uM | ALA4235137 | nM | ||||
3. | ALA4248974 | 19 | EC50 | = | 2 | nM | ALA4235136 | 8.70 | nM | Homo sapiens | ||
4. | ALA4248974 | 19 | IC50 | = | 10 | nM | ALA4235135 | 8.00 | nM | Homo sapiens | ||
5. | ALA4248974 | 19 | IC50 | = | 13 | nM | ALA4235134 | 7.89 | nM | Homo sapiens | ||
6. | ALA4248974 | 19 | CI | < | 1 | ALA4235142 | Homo sapiens | |||||
7. | ALA4248974 | 19 | CI | < | 1 | ALA4235143 | Homo sapiens | |||||
8. | ALA4248974 | 19 | CI | = | 0.75 | ALA4235144 | Homo sapiens | |||||
9. | ALA4248974 | 19 | CI | = | 0.68 | ALA4235145 | Homo sapiens | |||||
10. | ALA4248974 | 19 | CI | = | 0.97 | ALA4235146 | Homo sapiens | |||||
11. | ALA4248974 | 19 | CI | = | 0.72 | ALA4235147 | Homo sapiens | |||||
12. | ALA4248974 | 19 | INH | 0 | ALA4235148 | Not Active | % | Homo sapiens | ||||
13. | ALA4248974 | 19 | Stability | 0 | ALA4235132 | Stable | % | |||||
14. | ALA4248974 | 19 | Stability | 0 | ALA4235149 | Stable | % | |||||
15. | ALA4248974 | 19 | INH | 0 | ALA4235150 | Not Active | % | |||||
16. | ALA4248974 | 19 | F | = | 15 | % | ALA4235151 | % | Rattus norvegicus | |||
17. | ALA4248974 | 19 | Activity | = | 91.5 | % | ALA4235153 | % | Homo sapiens | |||
18. | ALA4248974 | 19 | Activity | = | 93.7 | % | ALA4235154 | % | Homo sapiens | |||
19. | ALA4248974 | 19 | Activity | = | 24.7 | mm3 | ALA4235155 | mm3 | Homo sapiens | |||
20. | ALA4248974 | 19 | Drug uptake | = | 0.2 | ug ml-1 | ALA4235156 | ug ml-1 |