| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4250253 | M2 | CLH | < | 3 | uL/min | ALA4234626 | uL/min | Homo sapiens | |||
| 2. | ALA4250253 | M2 | t1/2 | > | 400 | min | ALA4234627 | hr | ||||
| 3. | ALA4250253 | M2 | IC50 | = | 25 | uM | ALA4234628 | 4.60 | nM | Homo sapiens | ||
| 4. | ALA4250253 | M2 | EC50 | = | 2.11 | uM | ALA4234629 | 5.68 | nM | Homo sapiens | ||
| 5. | ALA4250253 | M2 | Activity | 0 | ALA4234629 | Dose-dependent effect | Homo sapiens | |||||
| 6. | ALA4250253 | M2 | Kd | = | 209.1 | nM | ALA4234630 | 6.68 | nM | Homo sapiens | ||
| 7. | ALA4250253 | M2 | K | = | 23 | 10'-3/s | ALA4234631 | 10'-3/s | Homo sapiens | |||
| 8. | ALA4250253 | M2 | K | = | 1.1 | 10'5/M/s | ALA4234632 | 10'5/M/s | Homo sapiens | |||
| 9. | ALA4250253 | M2 | t1/2 | = | 30.13 | s | ALA4234633 | hr | Homo sapiens | |||
| 10. | ALA4250253 | M2 | Papp | = | 0.3 | 10'-6 cm/s | ALA4234634 | 10'-6 cm/s | ||||
| 11. | ALA4250253 | M2 | logD | = | -0.05 | ALA4234635 | ||||||
| 12. | ALA4250253 | M2 | Activity | 0 | ALA4234636 | Not Determined | Homo sapiens | |||||
| 13. | ALA4250253 | M2 | Activity | 0 | ALA4234637 | Not Determined | Homo sapiens | |||||
| 14. | ALA4250253 | M2 | Activity | 0 | ALA4234638 | Not Determined | Homo sapiens | |||||
| 15. | ALA4250253 | M2 | Activity | = | 154 | % | ALA4234639 | % | Homo sapiens | |||
| 16. | ALA4250253 | M2 | Activity | = | 193 | % | ALA4234640 | % | Homo sapiens | |||
| 17. | ALA4250253 | M2 | EC50 | > | 40000 | nM | ALA4234621 | nM | Homo sapiens | |||
| 18. | ALA4250253 | M2 | EC50 | > | 40000 | nM | ALA4234641 | nM | Homo sapiens | |||
| 19. | ALA4250253 | M2 | EC50 | > | 40000 | nM | ALA4234642 | nM | Homo sapiens | |||
| 20. | ALA4250253 | M2 | EC50 | = | 353 | nM | ALA4234643 | 6.45 | nM | Homo sapiens |
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