| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4277551 | 14 | IC50 | = | 0.37 | uM | ALA4251893 | 6.43 | nM | Homo sapiens | ||
| 2. | ALA4277551 | 14 | IC50 | = | 0.95 | uM | ALA4251894 | 6.02 | nM | Homo sapiens | ||
| 3. | ALA4277551 | 14 | Ratio IC50 | = | 2.4 | ALA4251895 | ||||||
| 4. | ALA4277551 | 14 | CLH | = | 74 | microL/min/mg | ALA4251896 | mL.min-1.g-1 | ||||
| 5. | ALA4277551 | 14 | Therm_solubility | = | 96 | uM | ALA4251897 | nM | ||||
| 6. | ALA4277551 | 14 | CLH | = | 559 | microL/min/mg | ALA4251899 | mL.min-1.g-1 | ||||
| 7. | ALA4277551 | 14 | Fu | = | 0.037 | ALA4251900 | ||||||
| 8. | ALA4277551 | 14 | Cmax | = | 4.3 | uM | ALA4251901 | nM | Mus musculus | |||
| 9. | ALA4277551 | 14 | fCmax | = | 0.16 | uM | ALA4251902 | uM | Mus musculus | |||
| 10. | ALA4277551 | 14 | t1/2 | = | 3.1 | hr | ALA4251903 | hr | Mus musculus | |||
| 11. | ALA4277551 | 14 | IC50 | = | 18 | uM | ALA4251905 | 4.75 | nM | Homo sapiens | ||
| 12. | ALA4277551 | 14 | CL/F | = | 17 | L/hr/kg | ALA4251904 | mL.min-1.kg-1 | Mus musculus | |||
| 13. | ALA4277551 | 14 | Activity | 0 | ALA4251917 | Not Active | Mus musculus | |||||
| 14. | ALA4277551 | 14 | Ratio | = | 1.8 | ALA4251915 | ||||||
| 15. | ALA4277551 | 14 | Cp(f) | = | 0.82 | uM | ALA4251914 | uM | ||||
| 16. | ALA4277551 | 14 | Cp | = | 22 | uM | ALA4251913 | uM | ||||
| 17. | ALA4277551 | 14 | Activity | = | 76 | % | ALA4251911 | % | Mus musculus | |||
| 18. | ALA4277551 | 14 | Ratio | = | 1.5 | ALA4251910 | Homo sapiens | |||||
| 19. | ALA4277551 | 14 | Ratio | = | 1.1 | ALA4251909 | ||||||
| 20. | ALA4277551 | 14 | Papp | = | 36 | ucm/s | ALA4251908 | ucm/s |
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