# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4282356 | rac-12a; C149 | Drug metabolism | 0 | ALA4256881 | Metabolite_Detected | ||||||
2. | ALA4282356 | rac-12a; C149 | AUC | = | 294 | nmol.hr/ml | ALA4256875 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | Macaca fascicularis | ||
3. | ALA4282356 | rac-12a; C149 | t1/2 | = | 3 | hr | ALA4256869 | hr | Macaca fascicularis | |||
4. | ALA4282356 | rac-12a; C149 | Cmax | = | 55 | uM | ALA4256863 | nM | Macaca fascicularis | |||
5. | ALA4282356 | rac-12a; C149 | Tmax | = | 2 | hr | ALA4256857 | hr | Macaca fascicularis | |||
6. | ALA4282356 | rac-12a; C149 | IC50 | = | 2.1 | nM | ALA4256853 | 8.68 | nM | Homo sapiens |