| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4282387 | 27a | F | = | 98.1 | % | ALA4268597 | % | Rattus norvegicus | |||
| 2. | ALA4282387 | 27a | CL | = | 139.2 | ml/min.kg | ALA4268596 | mL.min-1.kg-1 | Rattus norvegicus | |||
| 3. | ALA4282387 | 27a | Cmax | = | 129.4 | ng/ml | ALA4268595 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 4. | ALA4282387 | 27a | Cmax | = | 72.1 | ng/ml | ALA4268594 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | Rattus norvegicus | ||
| 5. | ALA4282387 | 27a | Tmax | = | 5 | hr | ALA4268593 | hr | Rattus norvegicus | |||
| 6. | ALA4282387 | 27a | AUC | = | 1174.3 | ng.hr/ml | ALA4268592 | ng.hr.mL-1 | Rattus norvegicus | |||
| 7. | ALA4282387 | 27a | AUC | = | 239.42 | ng.hr/ml | ALA4268591 | ng.hr.mL-1 | Rattus norvegicus | |||
| 8. | ALA4282387 | 27a | t1/2 | = | 5 | hr | ALA4268590 | hr | Rattus norvegicus | |||
| 9. | ALA4282387 | 27a | t1/2 | = | 2.16 | hr | ALA4268589 | hr | Rattus norvegicus | |||
| 10. | ALA4282387 | 27a | logP | = | 2.98 | ALA4268588 | ||||||
| 11. | ALA4282387 | 27a | solubility | = | 20.47 | ug ml-1 | ALA4268587 | ug.mL-1 | ||||
| 12. | ALA4282387 | 27a | Activity | 0 | ALA4268586 | Dose-dependent effect | Mus musculus | |||||
| 13. | ALA4282387 | 27a | Activity | = | 1.56 | % | ALA4268585 | % | Mus musculus | |||
| 14. | ALA4282387 | 27a | Activity | = | 94.6 | % | ALA4268584 | % | Mus musculus | |||
| 15. | ALA4282387 | 27a | Activity | = | 6.99 | % | ALA4268583 | % | Mus musculus | |||
| 16. | ALA4282387 | 27a | Activity | = | 14.1 | % | ALA4268582 | % | Mus musculus | |||
| 17. | ALA4282387 | 27a | Activity | = | 76 | % | ALA4268581 | % | Mus musculus | |||
| 18. | ALA4282387 | 27a | Activity | = | 0 | % | ALA4268580 | % | Mus musculus | |||
| 19. | ALA4282387 | 27a | Activity | = | 16.4 | % | ALA4268579 | % | Mus musculus | |||
| 20. | ALA4282387 | 27a | Activity | = | 35.9 | % | ALA4268578 | % | Mus musculus |
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